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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

Potent and selective sst2 agonist CAS# 208706-12-1

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

Catalog No. BCC7364----Order now to get a substantial discount!

Product Name & Size Price Stock
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264: 5mg $702 In Stock
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264: 10mg Please Inquire In Stock
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264: 20mg Please Inquire Please Inquire
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264: 50mg Please Inquire Please Inquire
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264: 100mg Please Inquire Please Inquire
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264: 200mg Please Inquire Please Inquire
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264: 500mg Please Inquire Please Inquire
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264: 1000mg Please Inquire Please Inquire
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Quality Control of (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

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Chemical structure

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264

3D structure

Chemical Properties of (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

Cas No. 208706-12-1 SDF Download SDF
PubChem ID 9915239 Appearance Powder
Formula C33H41N5O2 M.Wt 539.71
Type of Compound N/A Storage Desiccate at -20°C
Solubility Soluble to 50 mM in DMSO and to 100 mM in ethanol
Chemical Name N-[(2R)-1-[[(1R,3S)-3-(aminomethyl)cyclohexyl]methylamino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]spiro[indene-1,4'-piperidine]-1'-carboxamide
SMILES C1CC(CC(C1)CNC(=O)C(CC2=CNC3=CC=CC=C32)NC(=O)N4CCC5(CC4)C=CC6=CC=CC=C56)CN
Standard InChIKey DAMXHAMKVXERLM-FVBCXUTKSA-N
Standard InChI InChI=1S/C33H41N5O2/c34-20-23-6-5-7-24(18-23)21-36-31(39)30(19-26-22-35-29-11-4-2-9-27(26)29)37-32(40)38-16-14-33(15-17-38)13-12-25-8-1-3-10-28(25)33/h1-4,8-13,22-24,30,35H,5-7,14-21,34H2,(H,36,39)(H,37,40)/t23-,24+,30+/m0/s1
General tips For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.
We recommend that you prepare and use the solution on the same day. However, if the test schedule requires, the stock solutions can be prepared in advance, and the stock solution must be sealed and stored below -20℃. In general, the stock solution can be kept for several months.
Before use, we recommend that you leave the vial at room temperature for at least an hour before opening it.
About Packaging 1. The packaging of the product may be reversed during transportation, cause the high purity compounds to adhere to the neck or cap of the vial.Take the vail out of its packaging and shake gently until the compounds fall to the bottom of the vial.
2. For liquid products, please centrifuge at 500xg to gather the liquid to the bottom of the vial.
3. Try to avoid loss or contamination during the experiment.
Shipping Condition Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other couriers with RT, or blue ice upon request.

Biological Activity of (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

DescriptionPotent and selective somatostatin sst2 receptor agonist (Ki values are 4, 537, 2480, 3614 and 5017 nM for cloned human sst2, sst1, sst4, sst3 and sst5 receptors respectively).

(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Dilution Calculator

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(1R,1'S,3'R/1R,1'R,3'S)-L-054,264 Molarity Calculator

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Preparing Stock Solutions of (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

1 mg 5 mg 10 mg 20 mg 25 mg
1 mM 1.8528 mL 9.2642 mL 18.5285 mL 37.0569 mL 46.3212 mL
5 mM 0.3706 mL 1.8528 mL 3.7057 mL 7.4114 mL 9.2642 mL
10 mM 0.1853 mL 0.9264 mL 1.8528 mL 3.7057 mL 4.6321 mL
50 mM 0.0371 mL 0.1853 mL 0.3706 mL 0.7411 mL 0.9264 mL
100 mM 0.0185 mL 0.0926 mL 0.1853 mL 0.3706 mL 0.4632 mL
* Note: If you are in the process of experiment, it's necessary to make the dilution ratios of the samples. The dilution data above is only for reference. Normally, it's can get a better solubility within lower of Concentrations.

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