Muscarinic Receptor
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
Products for Muscarinic Receptor
- Cat.No. Product Name Information
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BCC1470
CevimelineMuscarinic receptor agonist
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BCC1471
Cevimeline hydrochloride hemihydrateAgonist of muscarinic receptor (M1/M3)
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BCC1516
DarifenacinM3 receptor antagonist and antimuscarinic agents
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BCC2022
Umeclidinium bromideMAChR antagonist
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BCC4565
Biperiden HClMuscarinic receptor antagonist; some selectivity for M1
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BCC4567
Darifenacin HBr
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BCC4575
Aclidinium BromideLAMAs antagonist
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BCC4580
Solifenacin succinateMuscarinic receptor antagonist
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BCC4583
5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM)
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BCC4584
Fesoterodine Fumarate
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BCC4586
Tolterodine tartratePotent, non-selective muscarinic receptor antagonist
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BCC6164
VU 0365114Positive allosteric modulator of M5 receptors
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BCC6217
PTAC oxalateMuscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes
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BCC6627
Arecaidine but-2-ynyl ester tosylate
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BCC6628
Arecaidine propargyl ester tosylateMuscarinic agonist
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BCC6655
Nitrocaramiphen hydrochlorideMuscarinic antagonist, M1 > M2
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BCC6661
4-DAMPMuscarinic M3 antagonist
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BCC6682
W-84 dibromideStabilizer of cholinergic antagonist-receptor complexes
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BCC6707
5-MethylfurmethiodidePotent muscarinic agonist
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BCC6814
Oxotremorine sesquifumarateMuscarinic agonist
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BCC6920
Oxotremorine MMuscarinic agonist
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BCC6923
Pirenzepine dihydrochlorideSelective M1 muscarinic antagonist
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BCC6939
AF-DX 116Selective M2 antagonist
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BCC6946
Telenzepine dihydrochloridePotent, selective M1 antagonist
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BCC7024
AF-DX 384Potent M2/M4 antagonist
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BCC7042
McN-A 343Selective M1 muscarinic agonist
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BCC7061
(S)-(+)-Dimethindene maleateH1 antagonist. Also M2 muscarinic antagonist
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BCC7145
PD 102807Selective M4 antagonist
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BCC7263
DAU 5884 hydrochlorideM3 receptor antagonist
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BCC7314
AQ-RA 741Selective, high affinity M2 antagonist
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BCC7389
J 104129 fumaratePotent, selective M3 antagonist
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BCC7418
Zamifenacin fumarateSelective M3 antagonist
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BCC7427
Milameline hydrochlorideMuscarinic receptor agonist
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BCC7556
(+)-Muscarine iodideMuscarinic receptor agonist
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BCC7577
VU 10010
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BCC7729
VU 0238429Selective positive allosteric modulator of M5 receptors
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BCC7766
VU 0255035Highly selective muscarinic M1 antagonist
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BCC7907
VU 0357017 hydrochloridePositive allosteric modulator of M1 receptors