Products for Protease-Activated Receptors
- Cat.No. Product Name Information
-
BCC6281
Q94 hydrochloride
-
BCC6041
Parstatin (human)
-
BCC6042
Parstatin (mouse)
-
BCC7125
SCH 79797 dihydrochloride
SCH79797 dihydrochloride is a highly potent, selective nonpeptide protease activated receptor 1 (PAR1) antagonist. SCH79797 dihydrochloride inhibits binding of a high-affinity thrombin receptor-activating peptide to PAR1 with an IC50 of 70 nM and a Ki of 35 nM. SCH79797 dihydrochloride inhibits thrombin-induced platelet aggregation with an IC50 of 3 μM. SCH79797 dihydrochloride has antiproliferative and pro-apoptotic effects, and limits myocardial ischemia/reperfusion injury in rat hearts. SCH79797 dihydrochloride also potently prevents PAR1 activation in vascular smooth muscle cells, endothelial cells, and astrocytes.
-
BCC7392
APC 366
Tryptase inhibitor
-
BCC7734
FR 171113
-
BCC6279
FSLLRY-NH2
-
BCC7433
RWJ 56110
-
BCC5770
tcY-NH2
