Adenosine A2B Receptor
Adenosine A2B receptors are members of the adenosine receptor group of G-protein-coupled receptors that also includes A1, A2A and A3. A2B receptors display high expression levels in the cecum, colon and bladder, with lower levels in the lung, blood vessels and eye.
Products for Adenosine A2B Receptor
- Cat.No. Product Name Information/Activity
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BCC6197
BAY 60-6583
BAY 60-6583 is a potent and high-affinity agonist of adenosine A2B receptor (EC50 = 3 nM) over A1, A2A, and A3 receptors. BAY 60-6583 binds to mouse, rabbit, and dog A2BAR with Ki values of 750 nM, 340 nM and 330 nM, respectively. BAY 60-6583 has a cardioprotective effect in a myocardial ischemia model.
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BCC7163
CV 1808
53296-10-9
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BCC6237
LUF 5834
333962-91-7
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BCC7120
MRS 1706
MRS-1706 is a potent and selective adenosine A2B receptor inverse agonist. MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1 and A3 receptors respectively.
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BCC7473
MRS 1754
MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats.
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BCC7237
PSB 1115
152529-79-8
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BCC7598
PSB 603
1092351-10-4
