Apelin Receptor
Apelin-36, apelin-13 and [Pyr1]-apelin-13 are the predominant endogenous ligands for the apelin receptor (APJ) receptor. The APJ receptor and apelin peptides act as mediators of cardiovascular function, fluid homeostasis and adipocyte endocrine secretion.
Products for Apelin Receptor
- Cat.No. Product Name Information/Activity
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BCC7358
[Pyr1]-Apelin-13
[Pyr1]-Apelin-13 is a highly potent, selective endogenous apelin receptor (APJ) agonist.
![[Pyr1]-Apelin-13 chemical structure](/media/images/struct/BCC7358.png)
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BCC5959
Apelin-17 (human, bovine)
217082-57-0
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BCC5910
Apelin-36 (human)
252642-12-9
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BCC5911
Apelin-36 (rat, mouse)
230299-95-3
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BCC6278
ML 221
ML221 is a potent apelin (APJ) functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays.
