Glutamate (Metabotropic) Group I Receptor
Metabotropic glutamate (mGlu) group I receptors are members of the metabotropic class of glutamate receptors, which also includes mGlu group II and mGlu group III receptors. mGlu group I receptors are divided into two subtypes, mGlu1 and mGlu5.
Products for Glutamate (Metabotropic) Group I Receptor - Page 4
- Cat.No. Product Name Information/Activity
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BCC1777
MPEP Hydrochloride
MPEP hydrochloride is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype with IC50 of 36 nM.
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BCC1780
MTEP hydrochloride
MTEP hydrochloride is a potent, selective and non-competitive mGlu5 antagonist with an IC50 of 5 nM and a Ki of 16 nM. MTEP hydrochloride produces antiparkinsonian-like effects.
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BCC6119
NPS 2390
226878-01-9
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BCC6895
PHCCC
PHCCC is a Group I metabotropic glutamate receptor antagonist with EC 50 of 6 uM and a positive allosteric modulator of mGluR4. Also as a potent to antagonism for mGluR2 and mGluR8.
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BCC6971
SIB 1757
31993-01-8
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BCC7682
YM 202074
299900-84-8
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BCC5956
YM 230888
446257-23-4
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BCC7366
YM 298198 hydrochloride
1216398-09-2
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BCC7365
Desmethyl-YM 298198
1177767-57-5
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BCC6171
ADX 10059 hydrochloride
Negative allosteric modulator at mGlu<sub>5</sub>
