5-HT2C Receptor
Serotonin 5-HT2C receptors, previously known as 5-HT1C receptors, are located primarily in the choroid plexus, cortex, limbic system and basal ganglia. 5-HT2C receptors play a role in CSF volume regulation, thermoregulation, penile erection and anxiety.
Products for 5-HT2C Receptor
- Cat.No. Product Name Information/Activity
-
BCC1499
CP-809101 hydrochloride
CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively.
-
BCC5680
m-CPP hydrochloride
13078-15-4
-
BCC5925
DOI hydrochloride
42203-78-1
-
BCC5422
Eltoprazine hydrochloride
Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.
-
BCC7536
1-Methylpsilocin
1465-16-3
-
BCC6856
MK 212 hydrochloride
61655-58-1
-
BCC7718
Org 12962 hydrochloride
210821-63-9
-
BCC7285
PNU 22394 hydrochloride
15923-42-9
-
BCC7196
Ro 60-0175 fumarate
169675-09-6
-
BCC6849
SCH 23390 hydrochloride
SCH-23390 hydrochloride (R-(+)-SCH-23390 hydrochloride) is a potent and selective dopamine D1-like receptor antagonist with Kis of 0.2 nM and 0.3 nM for the D1 and D5 receptor, respectively. SCH-23390 hydrochloride is a potent and high efficacy human 5-HT2C receptor agonist with a Ki of 9.3 nM. SCH-23390 hydrochloride also binds with high affinity to the 5-HT2 and 5-HT1C receptors. SCH-23390 hydrochloride inhibits G protein-coupled inwardly rectifying potassium (GIRK) channels with an IC50 of 268 nM.
