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Cat.No. Product Name Information/Activity

BCC7603 alpha,beta-Methyleneadenosine 5'-triphosphate trisodium salt α,β-Methylene ATP trisodium, a phosphonic analog of ATP, is a P2X3 and P2X7 receptor ligand.

alpha,beta-Methyleneadenosine 5'-triphosphate trisodium salt chemical structure

BCC6918 2-Methylthioadenosine triphosphate tetrasodium salt 100020-57-3

2-Methylthioadenosine triphosphate tetrasodium salt chemical structure

BCC1317 A 438079 hydrochloride A 438079 (hydrochloride) is a potent, and selective P2X7 receptor antagonist with pIC50 of 6.9. A 438079 hydrochloride chemical structure

A 438079 hydrochloride chemical structure

BCC1322 A-740003 A-740003 is a potent, selective and competitive P2X7 receptor antagonist with IC50 values are 18 and 40 nM for rat and human P2X7 receptors, respectively. A-740003 chemical structure

BCC6198 A 804598 A-804598 is a CNS penetrant, competitive and selective P2X7 receptor antagonist with IC50s of 9 nM, 10 nM and 11 nM for mouse, rat and human P2X7 receptors, respectively. A 804598 chemical structure

BCC4290 A 839977 A 839977 is a P2X7 selective antagonist; it blocks BzATP-evoked calcium influx at recombinant human, rat and mouse P2X7 receptors (IC50 values are 20 nM, 42 nM and 150 nM respectively) and reduces inflammatory and neuropathic pain in animal models; the antihyperalgesic effects of P2X7 receptor blockade are mediated by blocking the release of IL-1beta. A 839977 chemical structure

BCC6005 AZ 10606120 dihydrochloride AZ10606120 dihydrochloride is a selective, high affinity antagonist for P2X7 receptor (P2X7R) at human and rat with an IC50 of ~10 nM. AZ10606120 dihydrochloride is little or no effect at other P2XR subtypes. AZ10606120 dihydrochloride has anti-depressant effects and reduces tumour growth. AZ 10606120 dihydrochloride chemical structure

AZ 10606120 dihydrochloride chemical structure

BCC7646 AZ 11645373 Potent and selective human P2X<sub>7</sub> antagonist AZ 11645373 chemical structure

BCC7717 5-BDBD 768404-03-1 5-BDBD chemical structure

BCC6815 Evans Blue tetrasodium salt Selective P2X purinergic antagonist,Evans Blue is a potent inhibitor of L-glutamate uptake via the membrane bound excitatory amino acid transporter (EAAT). Evans Blue tetrasodium salt chemical structure

Evans Blue tetrasodium salt chemical structure

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