5-HT1A Receptor
The serotonin 5-HT1A receptor was the first 5-HT receptor to be fully sequenced. 5-HT1A receptor binding sites are located primarily in limbic brain areas, notably the hypothalamus and cortical areas. The human gene encoding this receptor has been localized to chromosome 5.
Products for 5-HT1A Receptor
- Cat.No. Product Name Information/Activity
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BCC5034
Aripiprazole
Aripiprazole (OPC-14597) is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM.
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BCC7657
ATC 0175 hydrochloride
MCH<sub>1</sub> antagonist; also 5-HT<sub>2B</sub> antagonist and 5-HT<sub>1A</sub> partial agonist
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BCC5063
BMY 7378
5-HT<sub>1A</sub> partial agonist,BMY 7378 is a multi-targeted inhibitor of α2C-adrenoceptor and α1D-adrenoceptor with pKi of 6.54 and 8.2, respectively, and acts as a mixed agonist and antagonist for 5-HT1A receptor with pKi of 8.3.
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BCC6695
BP 554 maleate
Selective 5-HT<sub>1A</sub> agonist
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BCC6929
(R)-(+)-8-Hydroxy-DPAT hydrobromide
78095-19-9
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BCC6681
8-Hydroxy-DPAT hydrobromide
76135-31-4
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BCC6800
8-Hydroxy-PIPAT oxalate
1451210-48-2
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BCC7201
Ipsapirone
95847-70-4
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BCC6636
MDL 73005EF hydrochloride
102908-60-1
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BCC7165
Nemonapride
75272-39-8
