Sigma1 Receptor

σ 1 receptors are members of the σ family of receptors that also includes σ 2 receptors. They are distinguished from σ 2 receptors as they have high affinity and stereoselectivity for the (+)-isomers of pentazocine, SK&F 10047 and cyclazocine, and different subcellular localizations.

Products for Sigma1 Receptor - Page 2

Cat.No. Product Name Information/Activity
BCC6777 4-IBP 4-IBP is a selective σ1 agonist with a high level of affinity for the σ1 receptor (Ki = 1.7 nM) and a moderate affinity for the σ2 receptor (Ki = 25.2 nM) .
BCC5902 (+)-Igmesine hydrochloride 130152-35-1
BCC7429 PD 144418 oxalate PD 144418 is a highly affinity, potent and selective sigma 1 (σ1) receptor ligand (Ki values of 0.08 nM and 1377 nM for σ1 and σ2 respectively), devoid of any significant affinity for other receptors, ion channels and enzymes. PD 144418 shows potential antipsychotic activity.
BCC6784 N-[2-(Piperidinylamino)ethyl]-4-iodobenzamide 155054-42-5
BCC7450 TC 1 362512-81-0
BCC7251 SKF 83959 hydrobromide 67287-95-0