Products for Somatostatin Receptor
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BCC5945
BIM 23052
sst<sub>5</sub> agonist
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BCC6248
TT 232
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BCC5824
BIM 23056
sst receptor ligand
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BCC5913
CH 275
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BCC5823
CYN 154806
CYN 154806, a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively.
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BCC6010
Cortistatin 14
Cortistatin 14, human, rat (CST-14, human, rat), a neuropeptide with neuronal depressant and sleep modulating properties, can bind to all five cloned somatostatin receptors (SSTRs) and ghrelin receptor to exert its biological activities and co-exists with GABA within the cortex and hippocampus.
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BCC7361
NNC 26-9100
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BCC7364
(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
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BCC7220
L-803,087 trifluoroacetate
L-803087 is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM, which is > 280-fold higher than other somatostatin receptors. L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice.
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BCC7221
L-817,818
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BCC5300
Pasireotide
Pasireotide(SOM 230) is a stable cyclohexapeptide somatostatin mimic that exhibits unique high-affinity binding to human somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9 respectively).
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BCC5715
Somatostatin 1-28
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BCC7191
Seglitide
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BCC5643
Octreotide acetate
Octreotide is a somatostatin analog that binds to the somatostatin receptor, mainly subtypes 2, 3, and 5, increases Gi activity, and reduces intracellular cAMP production.
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BCC7693
Cyclosomatostatin
Non-selective sst receptor antagonist
