Products with Adrenergic receptor blockers Bioactivity

Explore BioCrick products associated with Adrenergic receptor blockers biological activity, including catalog numbers, product names and available bioactivity information.

Adrenergic receptor blockers Bioactivity Products

Cat. No. Product Name
BCN2262 Quinine HCl
1. Quinine HCl produces alpha-adrenergic blockade. 2. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
BCN5578 Isorauhimbine
1.3-Epi-alpha-yohimbine(Isorauhimbine) has alpha adrenoceptor blocking activities, has cardiovascular effects.
BCN5643 Stephanine
1. l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of 6.76. 2. Stephanine and crebanine have high inhibitory activity against gram-positive animal pathogenic bacteria, with MIC values of 0.078-0.312g/l, but low inhibitory activity against gram-negative animal pathogenic bacteria, they also inhibit hyphal growth of the plant pathogens Cercospora kaki. 3. Stephanine, pseudopalmatine , tetrahydropalmatine , and xylopinine show significant antiplasmodial activities with IC(50) ranged from 1.2 uM to 52.3 uM.
BCN5733 beta-Yohimbine
1. Beta-Yohimbine has anti-plasmodial and anti-malarial activity. 2. Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. 3. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor blocking activities, it has cardiovascular effects.
BCN6268 Yohimbine Hydrochloride
Yohimbine hydrochloride is an alpha 2-adrenoreceptor antagonist, blocking the pre- and postsynaptic alpha-2 adrenoreceptors and causing an increased release of noradrenaline and dopamine.It is an antagonist to xylazine hydrochloride-ketamine hydrochloride immobilization of white-tailed deer. Yohimbine has been used as a mydriatic and in the treatment of impotence. It is also alleged to be an aphrodisiac.

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