Products with Inhibitors bioactivity
| Cat.No. | Product Name |
|---|---|
| BCN6614 | Perilloxin |
| 1.Perilloxin possesses inhibitory activities against cyclooxygenase-1,with IC(50) values of 23.2 microM. | |
| BCN6635 | Beta-Peltoboykinolic acid |
| 1. Beta-Peltoboykinolic acid has in vitro protein tyrosine phosphatase 1B (PTP1B) inhibitory, it inhibits PTP1B with IC50 values of 5.2+/-0.5 microM. 2. Beta-Peltoboykinolic acid has cytotoxic activity. | |
| BCN6637 | 11-O-Galloylbergenin |
| 1. 11-O-Galloylbergenin shows significant analgesic activity at doses of 20 and 40 mg/kg against formalin test in rats, and it exhibits significant anti-inflammatory activity in carrageenan-induced paw edema model at doses of 10, 20 and 30 mg/kg. 2. 11-O-Galloylbergenin shows good antioxidant and antiplasmodial activities, the EC50 values are 7.45±0.2 ug/mL and 5.39±0.28 ug/mL in DPPH antioxidant assay and reducing power assay respectively, while IC50 value for antiplasmodial assay is less than 2.5 uM. 3. 11-O-Galloylbergenin shows significant urease inhibitory potential with IC50 value of 38.6±1.5 uM. | |
| BCN6670 | Ladanein |
| 1. Ladanein displays moderate (20-40 microM) activities against K562, K562R (imatinib-resistant), and 697 human leukemia cell lines . 2. Ladanein possesses free radicals DPPH and ABTS +.scavenging activity. 3. Ladanein is a phytochemicals inhibitor that is known to disrupt the interactions of core and other hepatitis C virus (HCV) proteins. | |
| BCN6680 | 2,3-Dihydrohinokiflavone |
| 1. 2,3-Dihydrohinokiflavone (IC50 =1.6uM) shows strong activity against Leishmania. 2. 2,3-Dihydrohinokiflavone is a suppressor of matrix metalloproteinases (MMPs) gene expression. | |
