Others Products Targets
- Other Nuclear Receptors (6)
- Vitamin D Receptor (10)
- Apelin Receptor (5)
- Thyrotropin-Releasing Hormone Receptor (1)
- Somatostatin (sst) Receptor (14)
- Progesterone Receptor (4)
- Parathyroid Hormone Receptor (1)
- PACAP Receptor (3)
- NPY Receptor (22)
- Natriuretic Peptide Receptor (4)
- Motilin Receptor (3)
- Mineralocorticoid Receptor (7)
- Melatonin Receptor (10)
- Melanocortin (MC) Receptor (17)
- Leptin Receptor (1)
- Kisspeptin Receptor (4)
- Insulin and Insulin-like Receptors (9)
- Gonadotropin-Releasing Hormone Receptor (3)
- Ghrelin Receptor (12)
- Galanin Receptor (11)
- Estrogen and Related Receptor (33)
- Calcitonin and Related Receptor (10)
- Bombesin Receptor (12)
- OX2 Receptor (4)
- OX1 Receptor (5)
- Secretin Receptor (1)
- Glucagon-Like Peptide 2 Receptor (2)
- Glucagon-Like Peptide 1 Receptor (7)
- Glucagon Receptor (3)
- Androgen Receptor (11)
- GIP Receptor (1)
- CRF2 Receptor (3)
- CRF1 Receptor (5)
- CCK2 Receptor (7)
- CCK1 Receptor (3)
- VIP Receptor (7)
- ETB Receptor (6)
- ETA Receptor (5)
- Angiotensin AT2 Receptor (3)
- Angiotensin AT1 Receptor (9)
Products for Others - Page 17
- Cat.No. Product Name Information/Activity
-
BCC7613
BMS 193885
Potent, competitive NPY Y<sub>1</sub> receptor antagonist
-
BCC5882
BVD 10
Highly selective NPY Y<sub>1</sub> receptor antagonist; devoid of Y<sub>4</sub> agonist activity
-
BCC7283
CGP 71683 hydrochloride
CGP71683 hydrochloride is a competitive neuropeptide Y5 receptor antagonist with a Ki of 1.3 nM, and shows no obvious activity at Y1 receptor (Ki, >4000 nM) and Y2 receptor (Ki, 200 nM) in cell membranes.
-
BCC6238
CYM 9484
CYM 9484 is a selective and highly potent neuropeptide Y (NPY) Y2 receptor antagonist with an IC50 value of 19 nM.
-
BCC6100
JNJ 5207787
JNJ-5207787 is a nonpeptidic, selective and penetrate the blood-brain barrier neuropeptide Y Y2 receptor (Y2) antagonist. JNJ-5207787 inhibits the binding of peptide YY (PYY) with pIC50s of 7.0 and 7.1 for human Y2 receptor and rat Y2 receptor, respectively. JNJ-5207787 is >100-fold selective versus human Y1, Y4, and Y5 receptors.
-
BCC7041
L-152,804
L 152804 is an orally active and selective neuropeptide Y Y5 receptor (NPY5-R) antagonist, with a Ki of 26 nM for hY5. L 152804 causes weight loss in diet-induced obese mice by modulating food intake and energy expenditure.
-
BCC7708
LU AA33810
304008-29-5
-
BCC7747
NPY 5RA972
439861-56-0
-
BCC7270
NTNCB hydrochloride
191931-56-3
-
BCC7284
PD 160170
181468-88-2
