Others - BioCrick

Cat.No. Product Name Information/Activity

BCC5860 6-Iodonordihydrocapsaicin Potent, competitive vanilloid receptor antagonist 6-Iodonordihydrocapsaicin chemical structure

BCC7031 5'-Iodoresiniferatoxin 535974-91-5 5'-Iodoresiniferatoxin chemical structure

BCC7668 JNJ 17203212 JNJ-17203212 is a novel and selective TRPV1 antagonist, with IC50 of 65 nM and 102 nM for human TRPV1 and rat TRPV1. JNJ 17203212 chemical structure

BCC5779 L-R4W2 206350-79-0 L-R4W2 chemical structure

BCC7770 RN 1734 RN-1734 is selective antagonist of the TRPV4 channel, completely antagonizes 4αPDD-mediated activation of TRPV4 with comparable, low micromolar IC50s for all three species (hTRPV4: 2.3 μM, mTRPV4: 5.9 μM, rTRPV4: 3.2 μM). RN-1734 clearly decreases the production of tumor necrosis factor α (TNF-α) and interleukin 1β (IL-1β) without altering the number of olig2-positive cells. RN 1734 chemical structure

BCC7128 SB 366791 SB-366791 is a potent , competitive and selective vanilloid receptor (VR1/TRPV1) antagonist with IC50 of 5.7±1.2 nM target: VR1/TRPV1 IC 50: 5.7±1.2 nM [1] SB-366791 produced a concentration-dependent inhibition of the response to capsaicin with an apparent pKb of 7.74±0.08. SB 366791 chemical structure

BCC7620 SB 452533 459429-39-1 SB 452533 chemical structure

BCN5564 alpha-Spinasterol α-Spinasterol, isolated from Spinacia oleracea, has antibacterial activity. α-Spinasterol is a transient receptor potential vanilloid 1 (TRPV1) antagonist, has anti-inflammatory, antidepressant, antioxidant and antinociceptive effects. α-Spinasterol inhibits COX-1 andCOX-2 activities with IC50 values of 16.17 μM and 7.76 μM, respectively. alpha-Spinasterol chemical structure

BCC2514 Tranilast Tranilast is an antiallergic agent. Tranilast chemical structure

BCC6114 MM-22 956605-71-3 MM-22 chemical structure

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