Mu-Opioid Receptors
The μ opioid receptor, (also known as OP3, MOP, MOR), is a member of the opioid family of G-protein-coupled receptors that also includes κ , δ and NOP receptors. Three splice variants of the receptor (designated μ 1, μ 2 and μ 3) have been characterized.
Products for Mu-Opioid Receptors
- Cat.No. Product Name Information/Activity
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BCC6958
DAMGO
DAMGO is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR.
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BCC1008
Endomorphin-1
Endomorphin 1, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.
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BCC5697
Endomorphin-2
Endomorphin 2, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.
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BCC6000
Fentanyl citrate
990-73-8
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BCC4380
Loperamide HCl
Loperamide (hydrochloride) (R-18553 (hydrochloride)) is an opioid receptor agonist. Loperamide hydrochloride is a selective and competitive
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BCC4920
Meptazinol HCl
Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]dihydromorphine binding with IC50 of 58 nM.
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BCC6090
Oxycodone hydrochloride
124-90-3
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BCC5864
PL 017
83397-56-2
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BCN6318
Sinomenine HCl
6080-33-7
-
BCC5684
Clocinnamox mesylate
117332-69-1
