GABAA Receptor
GABAA receptors are members of the Cys-loop family of ligand-gated ion channels and, along with GABAB receptors, are responsible for mediating the inhibitory effects of GABA. They are pentameric proteins, consisting of five subunits belonging to different families.
Products for GABAA Receptor - Page 6
- Cat.No. Product Name Information/Activity
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BCC1150
Etomidate
Etomidate(R-16659) is a GABAA receptors agonist, which is a short acting intravenous anaesthetic agent used for the induction of general anaesthesia.
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BCC4456
Flupirtine maleate
Flupirtine Maleate(D 9998) is a selective neuronal potassium channel opener that also has NMDA receptor antagonist properties.
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BCC7397
Ganaxolone
38398-32-2
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BCC7720
Indiplon
325715-02-4
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BCC7009
Loreclezole hydrochloride
Loreclezole, an antiepileptic compound, is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit containing receptors.
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BCC7984
MaxiPost
Flindokalner (BMS-204352) is a potassium channel modulator. Flindokalner is a positive modulator of all neuronal Kv7 channel subtypes expressed in HEK293 cells. Flindokalner is also a large conductance calcium-activated K channel (BKca) positive modulator. Flindokalner shows a negative modulatory activity at Kv7.1 channels (Ki=3.7 μM), and acts as a negative modulator of GABAA receptors. Flindokalner shows anxiolytic efficacy in vivo.
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BCC6167
Ocinaplon
96604-21-6
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BCC7470
Org 20599
156685-94-8
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BCC7452
17-PA
694438-95-4
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BCC7736
Pregnanolone
128-20-1
