Products with Inhibitors bioactivity

Cat.No. Product Name
BCN3453 1,3,5,6-Tetrahydroxyxanthone
1. 1,3,5,6-Tetrahydroxyxanthone can inhibit angiotensin-I-converting-enzyme activity in a dose-dependent manner. 2. 1,3,5,6-Tetrahydroxyxanthone shows moderate hepatoprotective activity with EC(50) values of 160.2 +/- 0.6 microM against tacrine-induced cytotoxicity in HepG2 cells.
BCN3461 Alisol G
1. Alisol G has hCE2 inhibitory effects.
BCN3468 Skimmianin
1. Skimmianine is a new inhibitor against the Leishmania APRT enzyme. 2. Skimmianine has a selective inhibitory effect on the 5-hydroxytryptamine-induced vasopressor responses of rats. 3, Skimmianine is a strong acetylcholinesterase (AChE) inhibitor. 4. Skimmianine has anti-inflammatory properties. 5. Skimmianine has leishmanicidal effect , it is thus a promising drug candidate for L. braziliensis due to its potent immunomodulatory activity.
BCN3477 Purpurin
Purpurin is one of the natural colorants extracted from madder roots and other Rubiaceae family plants. Purpurin is a novel specific inhibitor of Adipocyte-derived leucine aminopeptidase, it exhibits anti-angiogenic, antifungal, antibiotic, and antioxidative activities.
BCN3489 Methyl reserpate
1. Methyl reserpate and reserpinediol, derivatives that incorporate the alkaloid ring system, also competitively inhibit norepinephrine transport into chromaffin vesicles with Ki values of 38 +/- 10 nM and 440 +/- 240 nM, respectively.

Items 356 to 360 of 625 total