Products with
Inhibitors bioactivity
Cat.No.
|
Product Name
|
BCN3453 |
1,3,5,6-Tetrahydroxyxanthone
|
1. 1,3,5,6-Tetrahydroxyxanthone can inhibit angiotensin-I-converting-enzyme activity in a dose-dependent manner.
2. 1,3,5,6-Tetrahydroxyxanthone shows moderate hepatoprotective activity with EC(50) values of 160.2 +/- 0.6 microM against tacrine-induced cytotoxicity in HepG2 cells. |
BCN3461 |
Alisol G
|
1. Alisol G has hCE2 inhibitory effects. |
BCN3468 |
Skimmianin
|
1. Skimmianine is a new inhibitor against the Leishmania APRT enzyme.
2. Skimmianine has a selective inhibitory effect on the 5-hydroxytryptamine-induced vasopressor responses of rats.
3, Skimmianine is a strong acetylcholinesterase (AChE) inhibitor.
4. Skimmianine has anti-inflammatory properties.
5. Skimmianine has leishmanicidal effect , it is thus a promising drug candidate for L. braziliensis due to its potent immunomodulatory activity. |
BCN3477 |
Purpurin
|
Purpurin is one of the natural colorants extracted from madder roots and other Rubiaceae family plants. Purpurin is a novel specific inhibitor of Adipocyte-derived leucine aminopeptidase, it exhibits anti-angiogenic, antifungal, antibiotic, and antioxidative activities. |
BCN3489 |
Methyl reserpate
|
1. Methyl reserpate and reserpinediol, derivatives that incorporate the alkaloid ring system, also competitively inhibit norepinephrine transport into chromaffin vesicles with Ki values of 38 +/- 10 nM and 440 +/- 240 nM, respectively. |