Kainate Receptor
Kainate receptors are members of the ionotropic class of glutamate receptors, which also includes NMDA and AMPA receptors. Kainate receptors have been identified both pre- and post-synaptically. They contribute to excitatory postsynaptic currents in many regions of the CNS.
Products for Kainate Receptor
- Cat.No. Product Name Information/Activity
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BCC6940
ATPA
ATPA is a selective glutamate receptor GluR5 activator with EC50s of 0.66, 9.5, 1.4, 23, 32, 18, and 14 μM for GluR5wt, GluR5(S741M), GluR5(S721T), GluR5(S721T, S741M), GluR5(S741A), GluR5(S741L), and GluR5(S741V), respectively.
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BCC6586
Domoic acid
14277-97-5
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BCC6597
(S)-(-)-5-Iodowillardiine
140187-25-3
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BCC6572
Kainic acid
Kainic acid is a potent agonist at excitatory amino acid receptor subtypes in the CNS.
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BCC7297
MNI caged kainic acid
1315378-75-6
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BCC6840
SYM 2081
SYM 2081 is a high-affinity ligand and potent, selective agonist of kainate receptors, inhibits [3H]-kainate binding with an IC50 of 35 nM, almost 3000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively.
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BCC7462
ACET
936095-50-0
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BCC6569
CNQX
CNQX (FG9065) is a potent AMPA/kainate receptor antagonist.
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BCC6908
CNQX disodium salt
479347-85-8
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BCC6815
Evans Blue tetrasodium salt
Selective P2X purinergic antagonist,Evans Blue is a potent inhibitor of L-glutamate uptake via the membrane bound excitatory amino acid transporter (EAAT).
