Products with
Antagonists bioactivity
Cat.No.
|
Product Name
|
BCN1062 |
Pseudoginsenoside F11
|
Pseudoginsenoside F11, a novel partial PPAR γ agonist, can promote adiponectin oligomerization and secretion in 3T3-L1 adipocytes and inhibit obesity-linked phosphorylation of PPAR γ at Ser-273 by Cdk5. It possesses significant neuroprotective activity, has been demonstrated to antagonize the learning and memory deficits induced by scopolamine, morphine and methamphetamine in mice; it also antagonizes the development of analgesia tolerance to morphine and blocks the development of morphine-induced behavioral sensitization via its effect, at least partially, on the glutamatergic system in the mPFC. |
BCN1187 |
Isohyenanchin
|
1. Isohyenanchin is a weak antagonist of ionotropic GABA receptors.
2. Isohyenanchin is the potent antagonist of RDLac homo-oligomers. |
BCN1232 |
DL-5-Hydroxytryptophan
|
5-Hydroxytryptophan (5-HTP) is the precursor of serotonin , has been widely used as a dietary supplement to raise serotonin level, it is an effective drug against depression, insomnia, obesity, chronic headaches, etc. 5-HTP supplementation can inhibit endothelial serotonylation, leukocyte recruitment, and allergic inflammation, it also can reduce the symptoms of anxiety/depression of that patients with allergy/asthma. 5-HTP
may be involved in inducing the female to stay in copula and delay egg-laying to prevent re-mating of the female. |