Products with Antagonists Bioactivity

Explore BioCrick products associated with Antagonists biological activity, including catalog numbers, product names and available bioactivity information.

Cat. No.	Product Name
BCN6578	Piperenone
1. Piperenone is an insect antifeeding substance. 2. Piperenone has anti-platelet-activating factor(PAF) activities, it is a PAF-acether antagonist.
BCN6632	(-)-Corlumine
1. Corlumine exhibits spasmolytic and GABA antagonist activity.
BCN6706	Yangambin
1. Yangambin is a selective antagonist of the cardiovascular effects of platelet activating factor (PAF) and therefore constitutes a potential therapeutic agent in different shock states where abnormal PAF release is supposed to play an important role. 2. Yangambin has central nervous system activity, it presents a depressant activity in the open field, forced swimming and pentobarbital sleeping time tests. 3. Yangambin has hypotensive effect, which is probably due to a peripheral vasodilatation that involves, at least, the inhibition the Ca2+ influx through voltage-gated Ca2+ channels.
BCN6785	Triptinin B
1. Triptinin A and triptinin B are leukotriene D4 antagonist constituents.
BCN6791	Cytosporone B
Cytosporone B is a naturally occurring agonist for Nur77, it also is a Salmonella pathogenicity island 1 (SPI-1)-inhibitor, it may have potential in drug development against antibiotic-resistant Salmonella. Cytosporone B can elevate blood glucose levels in fasting C57 mice, an effect that is accompanied by induction of multiple genes involved in gluconeogenesis. Cytosporone B can inhibit transforming growth factor-b (TGF-β)-induced contraction of human corneal fibroblasts (HCFs), likely as a result of its attenuation of the up-regulation of α-SMA expression.

Antagonists Bioactivity Products