Others Products Targets
- Other Nuclear Receptors (6)
- Vitamin D Receptor (10)
- Apelin Receptor (5)
- Thyrotropin-Releasing Hormone Receptor (1)
- Somatostatin (sst) Receptor (14)
- Progesterone Receptor (4)
- Parathyroid Hormone Receptor (1)
- PACAP Receptor (3)
- NPY Receptor (22)
- Natriuretic Peptide Receptor (4)
- Motilin Receptor (3)
- Mineralocorticoid Receptor (7)
- Melatonin Receptor (10)
- Melanocortin (MC) Receptor (17)
- Leptin Receptor (1)
- Kisspeptin Receptor (4)
- Insulin and Insulin-like Receptors (9)
- Gonadotropin-Releasing Hormone Receptor (3)
- Ghrelin Receptor (12)
- Galanin Receptor (11)
- Estrogen and Related Receptor (33)
- Calcitonin and Related Receptor (10)
- Bombesin Receptor (12)
- OX2 Receptor (4)
- OX1 Receptor (5)
- Secretin Receptor (1)
- Glucagon-Like Peptide 2 Receptor (2)
- Glucagon-Like Peptide 1 Receptor (7)
- Glucagon Receptor (3)
- Androgen Receptor (11)
- GIP Receptor (1)
- CRF2 Receptor (3)
- CRF1 Receptor (5)
- CCK2 Receptor (7)
- CCK1 Receptor (3)
- VIP Receptor (7)
- ETB Receptor (6)
- ETA Receptor (5)
- Angiotensin AT2 Receptor (3)
- Angiotensin AT1 Receptor (9)
Products for Others - Page 6
- Cat.No. Product Name Information/Activity
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BCC7062
PPT
Propyl pyrazole triol (PPT) is a selective estrogen receptor alpha (ERα) agonist. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 410 times higher compared with estrogen receptor beta (ERβ: 0.12%).
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BCC7669
WAY 200070
WAY-200070 is a selective estrogen receptor β (ERRβ) agonist with an IC50 of 2.3 nM.
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BCC1081
Fulvestrant
Fulvestrant (ICI 182780) is a pure antiestrogen and a potent estrogen receptor (ER) antagonist with an IC50 of 9.4 nM. Fulvestrant effectively inhibits the growth of ER-positive MCF-7 cells with an IC50 of 0.29 nM. Fulvestrant also induces autophagy and apoptosis and has antitumor efficacy.
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BCC7225
MPP dihydrochloride
MPP dihydrochloride is a highly selective estrogen receptor alpha (ERα) antagonist. MPP dihydrochloride reduces the ratio of p-ERα/ERα.
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BCC7447
PHTPP
PHTPP is a selective ERβ antagonist.
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BCC5121
XCT790
XCT-790 is a potent and selective inverse agonist for ERRα with an IC50 value of 0.37 μM. XCT-790 induces cell death in chemotherapeutic resistant cancer cells. XCT-790 (Compound 12) is inactive against ERRγ and the estrogen receptors ERα and ERβ.
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BCC7272
ZK 164015
177583-70-9
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BCC1412
Bazedoxifene acetate
Bazedoxifene acetate (TSE-424 acetate) is a third generation selective estrogen receptor modulator (SERM) with IC50s of 26 and 99 nM for ERα and ERβ, respectively.
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BCC7839
Cyclofenil
Cyclofenil is a selective estrogen receptor modulator and an ovulation-inducing agent. Cyclofenil shows an inhibitory effect on dengue virus replication in Vero cells with an EC50
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BCC6015
(Z)-4-Hydroxytamoxifen
4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM).
