Products with
Anticholinesterase bioactivity
Cat.No.
|
Product Name
|
BCN5523 |
Dipterocarpol
|
1. Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng.
2. Dipterocarpol A and hopeahainol A show moderate acetylcholinesterase inhibitory activity with IC50 values of 8.28 uM and 11.28 uM, respectively. |
BCN5705 |
1,3,5-Trihydroxy-4-prenylxanthone
|
1. 1,3,5-Trihydroxy-4-prenylxanthone is a relatively potent inhibitor of phosphodiesterase type 5 (PDE5), with an IC50 value of 3.0 μM.
2. 1,3,5-Trihydroxy-4-prenylxanthone inhibits LPS-induced NF-κB and AP-1 activations by interfering with the posttranslational modification (phosphorylation and/or ubiquitinylation) of IRAK-1 in the cell membrane to impede TAK1-mediated activation of IKK and MAPKs signal transduction.
3. 1,3,5-Trihydroxy-4-prenylxanthone shows in vitro inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE), with IC50 values of 56.3plusmn;0.4 and 46.0plusmn;0.3 M, respectively. |
BCN6033 |
Niloticin
|
1. Niloticin can be used as a potential natural mosquitocide, it shows strong larvicidal and pupicidal activities, and shows good mosquitocidal activity against Ae. aegypti.
2. Niloticin can be used against the larvae of A. aegypti as an effective acetylcholinesterase (AChE) inhibitor. |
BCN6158 |
2',4'-Dihydroxy-3',6'-dimethoxychalcone
|
1. 2',4'-Dihydroxy-3',6'-dimethoxychalcone has cytotoxic activities against cancer cells.
2. 2',4'-Dihydroxy-3',6'-dimethoxychalcone has anti-inflammatory activity and
anti-cholinesterase activity, it has significant NO inhibitory activity. |
BCN6209 |
Lycoclavanol
|
1. Lycoclavanol exhibits acetylcholinesterase inhibition activity. |