Products with
Anticholinesterase bioactivity
Cat.No.
|
Product Name
|
BCN1946 |
Hyoscyamine
|
Hyoscyamine is an AChR inhibitor with IC50 of 7.5 nM, it is widely used in medicine due to its anticholinergic activity. Hyoscyamine could be used to reduce abdominal discomfort and colonic spasm during a barium enema. |
BCN1953 |
Heleurine
|
1. Heleurine, platyphylline, supinine and cynaustraline are more potent in antagonizing responses to acetylcholine and carbachol than responses to histamine. |
BCN1980 |
Heliosupine
|
1. Heliosupine, heliosupine N-oxide, 3 ′-O-acetylheliosupine N-oxide,and 7-O-
angeloylechinatine N-oxide show inhibition activity against the acetylcholinesterase(AChE), with IC50 0.53-0.60 mM.
2. Heliosupine can deter feeding by the polyphagous larvae of Spodoptera exigua. |
BCN2098 |
Spectabiline
|
1. Spectabiline, monocrotaline, sarracine, lasiocarpine, 7-angelylheliotridine, heliotrine and senecionine have similar antagonistic potencies against responses to both acetylcholine and histamine.
2. Spectabiline shows tumor-inhibitory properties against one or more test tumors. |
BCN2669 |
Corydine
|
1. Corydine shows antimicrobial activity.
2. Corydine shows antineoplastic activity.
3. Corydine is the adrenolytic and weak cholinergic agent.
4. Corydine shows irritant and respiratory stimulant and CNS depressant activities .
5. Injected intravenously in rabbits corydine produced an initial fall in blood pressure followed by a return to normal or above normal. |