Hot Natural Products & Bioactive Compounds
BioCrick offers high-purity natural products and bioactive compounds for scientific research. Our natural product collection includes compounds derived from plants, microorganisms and other biological sources and is widely used in pharmacological, biochemical and drug discovery research.
Natural products remain an important source of bioactive molecules and drug leads. BioCrick provides researchers with high-quality natural product compounds together with catalog numbers, product information and biological activity data.
Hot Products from BioCrick
Showing 2321 - 2328 of 9359 hot products
| Catalog No. | Product Name |
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| BCC6876 | RS 79948 hydrochloride |
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<span class='symbol'>α</span><sub>2</sub>-adrenoreceptor antagonist (K<sub>d</sub> values are; 0.18, 0.19 and 0.42 nM for <span class='symbol'>α</span><sub>2B</sub> <span class='symbol'>α</span><sub>2C</sub> and <span class='symbol'>α</span><sub>2A</sub>, respectively in rat).
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| BCC6877 | RS 56812 hydrochloride |
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A highly potent and selective 5-HT3 partial agonist, with a pKi at 5-HT3 receptors in rat brain of 9.6, and greater than 1000-fold selectivity over a wide range of other neurotransmitter receptors.
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| BCC6878 | RS 67506 hydrochloride |
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A potent and selective 5-HT4 partial agonist, with a pKi of 8.8 at 5-HT4 sites in guinea pig striatum, but < 6.0 at several other receptors including 5-HT1A, 1D, 2A, 2C, D1, D2 and M1-3. It is active in vivo and has an intrinsic activity compared to 5-HT of 0.6.
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| BCC6879 | Isamoltane hemifumarate |
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5-HT<sub>1B</sub> antagonist, approximately 30-fold selective over 5-HT<sub>1A</sub>. Also possesses affinity for <span class='symbol'>β</span>-adrenergic receptors.
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| BCC6880 | Cyanopindolol hemifumarate |
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5-HT<sub>1A/1B</sub> antagonist with roughly equal affinity at each receptor; also a <span class='symbol'>β</span>-adrenoceptor antagonist.
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| BCC6881 | Pindolol |
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5-HT<sub>1A/1B</sub> receptor antagonist, with roughly equal affinity for each subtype. A partial agonist at mouse and human <span class='symbol'>β</span><sub>3</sub>-adrenoceptors. (<em>S</em>)-(-)-Pindolol also available.
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| BCC6882 | Spiperone hydrochloride |
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5-HT2A serotonin and selective D2-like dopamine receptor antagonist (Ki values are 0.06, 0.6, 0.08, ~ 350, ~ 3500 nM for D2, D3, D4, D1 and D5 receptors respectively). Antipsychotic.
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| BCC6883 | AH 11110 hydrochloride |
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A subtype-selective ligand for the <span class='symbol'>α</span><sub>1B</sub>-adrenoceptor. The pK<sub>i</sub> values for binding to rat fibroblast cell membranes expressing <span class='symbol'>α</span><sub>1B</sub> (hamster), <span class='symbol'>α</span><sub>1A</sub> (bovine) and <span class='symbol'>α</span><sub>1D</sub> (rat) are 7.1, 5.59, and 5.68 respectively. Appears to be non-selective between <span class='symbol'>α</span><sub>1</sub> subtypes and <span class='symbol'>α</span><sub>2</sub> receptors in smooth muscle preparations.
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