GPCR/G protein Compound Library

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GPCR/G protein Compound Library A unique collection of 756 natural compounds inhibitors/regulators for drug development and GPCR research/screening.

Catalog No. BCL0005

Size	Price	Stock
30 μL/well (10 mM solution)	Get quote	In-stock
30 μL/well (10 mM solution)	Get quote	In-stock
50 μL/well (10 mM solution)	Get quote	In-stock
100 μL/well (10 mM solution)	Get quote	In-stock
250 μL/well (10 mM solution)	Get quote	In-stock

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Description & Advantages

The products in the BioCrick screening libraries are all from plants.
The biological activities or pharmacological activities of all the BioCrick products are derived from the databases of all over the world the latest literatures, patent reports and clinical validation, you can according to the product manuals on our website to access the relevant literatures, hope that our informations can give some inspirations and help to your research.
The collections of unique natural products, which include antioxidants, anti-inflammatory, antibacterial, anticancer, and ect. Can be used for high throughput screening (HTS) and high content screening (HCS), is to help you carry out new drug screening, the emergence of new indications and other professional tools.
Available in stock with overnight delivery and free shipping over $500
A valuable tool for chemical genomics, epigenetic target identification in pharmacogenomics, and other biological applications.
Potent, selective and cell-permeable in inhibiting or activating target molecules
Bioactivity and safety confirmed by preclinical research and clinical trials.
Detailed files describing potency, selectivity and applications etc.
Structurally diverse, medicinally active, and cell permeable.
NMR and HPLC validated to ensure the highest purity.

Storage and Shipping Information

Form	Pre-dissolved DMSO solutions	Stability	-20°C: 12 months -80°C: 24 months
Packaging	96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode.
General tips	For obtaining a higher solubility , please warm the tube at 37°C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.
Shipping Condition	Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request

Contents of GPCR/G protein Compound Library

Plate layout: BCL0005

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	CP-945598 HCl	GW9508	Ramelteon	Macitentan	Ki16425	Plerixafor (AMD3100)	(R,R)-Formoterol	5-Iodotubercidin	AH 6809	AM095	Empty
b	Empty	AM-095 free base	AM630	AM966	AMD-070	AMD-070 hydrochloride	Anamorelin	Anamorelin Fumarate	Anamorelin hydrochloride	Atrasentan	Atrasentan hydrochloride	Empty
c	Empty	Avosentan	BAN ORL 24	Calcium-Sensing Receptor Antagonists I	Capadenoson	CCG-63802	CCG-63808	CGS 21680	Cinacalcet	CPPHA	Desmopressin	Empty
d	Empty	Desmopressin Acetate	Dipraglurant	Exendin-4	glucagon receptor antagonists 1	glucagon receptor antagonists 2	glucagon receptor antagonists 3	Glucocorticoid receptor agonist	GPR120 modulator 1	GPR120 modulator 2	GW-1100	Empty
e	Empty	HOKU-81	Ibutamoren Mesylate	INCB 3284 dimesylate	INCB3344	INCB8761(PF-4136309)	Indacaterol	JWH 073	Laropiprant	LUF6000	LY341495	Empty
f	Empty	MBX-2982	Medetomidine	mGlu2 agonist	MK 0893	MK-0812	MK-2894	MK-2894 sodium salt	MK-4305	MK-6892	MPEP Hydrochloride	Empty
g	Empty	MTEP hydrochloride	Nepicastat	NPS-2143 hydrochloride	ONO-AE3-208	Orteronel	Otenabant	PB-22	PD 123319 ditrifluoroacetate	Pentostatin	PF-543	Empty
h	Empty	Preladenant	Reparixin	Reparixin L-lysine salt	Rimonabant hydrochloride	RS 504393	Salmefamol	SB-408124 Hydrochloride	SCH 527123	SCH 563705	Setiptiline	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	Setiptiline maleate	sitaxsentan	SRT3109	SRT3190	TAK-700 salt	Talnetant hydrochloride	Taranabant	Tozadenant	TUG-770	Verlukast	Empty
b	Empty	Methylprednisolone	Tranilast	Zibotentan (ZD4054)	AM1241	TAK-875	Conivaptan HCl	GSK1292263	Istradefylline (KW-6002)	L-Glutamine	Mirabegron (YM178)	Empty
c	Empty	UNBS 5162	Vilanterol	Vilanterol trifenatate	AVE 0991	Detomidine	Alfuzosin	Prazosin	Tizanidine	L-(-)-α-Methyldopa hydrochloride	AHU-377(Sacubitril)	Empty
d	Empty	Azilsartan medoxomil monopotassium	Losartan	Tranilast Sodium	SCH 546738	NBI-74330	GPR40 Activator 1	GSK962040 hydrochloride	MCOPPB trihydrochloride	S1RA	S1RA hydrochloride	Empty
e	Empty	TAK-700 R-form	Levalbuterol tartrate	Doxazosin	AVE 0991 sodium salt	Perindopril	Betamethasone hydrochloride	Beclomethasone dipropionate	SB-334867	Prasugrel hydrochloride	Prasugrel Maleic acid	Empty
f	Empty	Siramesine	CGS 21680 HCl	DL-Adrenaline	Epinephrine HCl	Terbutaline Sulfate	Tolazoline HCl	Acebutolol HCl	Adrenalone HCl	Dexmedetomidine	Maprotiline HCl	Empty
g	Empty	Naphazoline HCl	Nebivolol	Phenoxybenzamine HCl	Propranolol HCl	Ritodrine HCl	Tetrahydrozoline HCl	Xylazine HCl	Betaxolol	Cisatracurium Besylate	Detomidine HCl	Empty
h	Empty	Epinephrine Bitartrate	Ivabradine HCl	Naftopidil	Phentolamine Mesylate	Terazosin HCl	Naftopidil DiHCl	Sotalol	Indacaterol Maleate	Synephrine HCl	Cinacalcet HCl	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	NPS-2143	BML-190	Org 27569	AM251	GW842166X	Rimonabant	Plerixafor 8HCl (AMD3100 8HCl)	WZ811	Mifepristone	Bosentan Hydrate	Empty
b	Empty	OC000459	Ki16198	MPEP	VU 0357121	CTEP (RO4956371)	Bosentan	Eprosartan Mesylate	Methyldopa	Montelukast Sodium	AdipoRon	Empty
c	Empty	Betamethasone	Budesonide	Cortisone acetate	Dexamethasone acetate	Nedaplatin	Prednisolone	Zafirlukast	Meprednisone	Fluticasone propionate	Bimatoprost	Empty
d	Empty	Alprostadil	Desonide	Ticlopidine HCl	Ticagrelor	MRS 2578	PF-05212384 (PKI-587)	Azilsartan Medoxomil	SKI II	Mozavaptan	Tolvaptan	Empty
e	Empty	BAF312 (Siponimod)	Almorexant	Almorexant hydrochloride	Guanfacine	AMD 3465	AMD 3465 hexahydrobromide	Dihydroergotamine mesylate	Ciclesonide	Misoprostol	Sarpogrelate hydrochloride	Empty
f	Empty	Ramosetron Hydrochloride	Kobe0065	kobe2602	Pasireotide	Atosiban	AL 8810	AZD1283	APD668	INT-777	PSN632408	Empty
g	Empty	Eltoprazine	Eltoprazine hydrochloride	RU 24969	Bambuterol	LPA2 antagonist 1	Labetalol HCl	RG7090	LCZ696	K-Ras G12C-IN-1	K-Ras G12C-IN-2	Empty
h	Empty	K-Ras G12C-IN-3	Fimasartan	K-Ras(G12C) inhibitor 12	ML224	Methylprednisolone Sodium Succinate	Octreotide acetate	2-Methyl-5-hydroxytryptamine hydrochloride	SB 203186 hydrochloride	GR 46611	m-CPP hydrochloride	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	MRS 2179 tetrasodium salt	Nociceptin	RS 67333 hydrochloride	RS 39604 hydrochloride	Methysergide maleate	[Phe1Ψ(CH2-NH)Gly2]Nociceptin(1-13)NH2	Nocistatin (bovine)	NocII	Bombesin	CGRP (rat)	Empty
b	Empty	Somatostatin 1-28	CGRP 8-37 (rat)	[Ac-Tyr1,D-Phe2]GRF 1-29, amide (human)	CGRP 8-37 (human)	VIP (guinea pig)	PACAP 1-27	Nocistatin (human)	Ac-RYYRIK-NH2	Nociceptin (1-7)	[Nphe1]Nociceptin(1-13)NH2	Empty
c	Empty	Nociceptin (1-13)NH2	SB 200646 hydrochloride	SB 204070	MRS 1334	[Ala11,22,28]VIP	Ac-RYYRWK-NH2	Galanin (1-15) (porcine, rat)	Galanin (2-29) (rat)	tcY-NH2	UFP-101	Empty
d	Empty	[(pF)Phe4]Nociceptin(1-13)NH2	[Arg14,Lys15]Nociceptin	[Orn8]-Urotensin II	2-Methylthioadenosine diphosphate trisodium salt	Urotensin II (human)	NECA	BAM (8-22)	Hemopressin (rat)	GRP (porcine)	GRP (human)	Empty
e	Empty	HS 014	HS 024	BIM 23127	CYN 154806	BIM 23056	Neuromedin C (porcine)	VIP (6-28) (human, rat, porcine, bovine)	Neuromedin N (rat, mouse, porcine, canine)	Neuromedin B (porcine)	Neurotensin	Empty
f	Empty	[D-Phe12]-Bombesin	Kinetensin (human)	Litorin	[D-Lys3]-GHRP-6	L-670,596	JMV 449	BWX 46	PHM 27 (human)	GIP (human)	Galnon	Empty
g	Empty	Oxyntomodulin	Xenin 8	MRS 2365	MRS 2279	MRS 2500 tetraammonium salt	BVD 10	GIP (1-39)	Motilin (human, porcine)	Tabimorelin hemifumarate	Bombinakinin-GAP	Empty
h	Empty	Bombinakinin M	ABT 702 dihydrochloride	DAPTA	Apelin-36 (human)	Apelin-36 (rat, mouse)	Obestatin (rat)	CH 275	UFP 803	DOI hydrochloride	Galanin (1-29) (rat, mouse)	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	M617	AR-M 1896	Bay 55-9837	BIM 187	BIM 189	SB 265610	SB 258719 hydrochloride	BX 513 hydrochloride	SC 51322	BIM 23052	Empty
b	Empty	DOB hydrochloride	SB 242084	[Des-octanoyl]-Ghrelin (rat)	Apelin-17 (human, bovine)	Galanin (porcine)	α-CGRP (human)	[Nle4,D-Phe7]-α-MSH	HOE 140	Cortistatin-8	[D-p-Cl-Phe6,Leu17]-VIP	Empty
c	Empty	HU 308	[Ala2,8,9,11,19,22,24,25,27,28]-VIP	d[Leu4,Lys8]-VP	[Orn5]-URP	Lys-[Des-Arg9]Bradykinin	R 892	Lys-Bradykinin	[Phe8Ψ(CH-NH)-Arg9]-Bradykinin	Sar-[D-Phe8]-des-Arg9-Bradykinin	BIM 23042	Empty
d	Empty	AR-C 66096 tetrasodium salt	CART (55-102) (rat)	CART (55-102) (human)	CART (62-76) (rat, human)	Cortistatin 14	(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin	R 715	Amylin	AC 187	SHU 9119	Empty
e	Empty	[D-Phe12,Leu14]-Bombesin	γ1-MSH	JKC 363	[Ala17]-MCH	MCL 0020	ACTH (1-39)	BX 471	SB 243213 dihydrochloride	Parstatin (human)	Parstatin (mouse)	Empty
f	Empty	CRSP-1	C 021 dihydrochloride	Lys-γ3-MSH	M 1145	SB 328437	Teijin compound 1	Hemopressin (human, mouse)	MCH (human, mouse, rat)	Orphanin FQ (1-11)	PSB 0739	Empty
g	Empty	JNJ 5207787	MRE 3008F20	8-Aminoadenine	MM-22	GSK 9027	KW 3902	MS 245 oxalate	SB 297006	MRS 2957 triethylammonium salt	TC-C 14G	Empty
h	Empty	TC-MCH 7c	5-OMe-UDP trisodium salt	26RFa	TC-G 1004	Psilocin	YE 120	AT 1015	EMD 281014 hydrochloride	BAY 60-6583	DV 7028 hydrochloride	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	SHA 68	CS 2100	IT1t dihydrochloride	TUG 891	LUF 5834	CYM 9484	MK 1903	TT 232	SB 706375	SB 611812	Empty
b	Empty	CYM 50260	CYM 50308	PU 02	LP 20 hydrochloride	TC-G 1006	ML 221	FSLLRY-NH2	Q94 hydrochloride	COR 170	BETP	Empty
c	Empty	Org 37684	PF 04418948	LUF 6283	CYM 5541	PG 106	CYM 50769	CID 16020046	ANQ 11125	PG 931	CTCE 9908	Empty
d	Empty	AMG837	Regadenoson	Rolapitant	ELN441958	Carteolol HCl	Metoprolol Succinate	Ozanimod (RPC1063)	N-Acetyltryptamine	DPCPX	m-Chlorophenylbiguanide hydrochloride	Empty
e	Empty	6-Chloromelatonin	5-Carboxamidotryptamine maleate	Cinanserin hydrochloride	Dihydroergocristine mesylate	1,3-Dipropyl-8-phenylxanthine	4F 4PP oxalate	MR 16728 hydrochloride	α-Methyl-5-hydroxytryptamine maleate	N-Methylquipazine dimaleate	PCA 4248	Empty
f	Empty	3-MPPI	Methiothepin maleate	PRE-084 hydrochloride	Metergoline	Quipazine dimaleate	Spiroxatrine	MDL 72222	3-AQC	2-Phenylmelatonin	RS 23597-190 hydrochloride	Empty
g	Empty	2-[1-(4-Piperonyl)piperazinyl]benzothiazole	2-Iodomelatonin	PG-9 maleate	SM-21 maleate	MDL 11,939	Luzindole	Oleamide	Palmitoylethanolamide	GR 135531	MK 212 hydrochloride	Empty
h	Empty	Zaprinast	1-Phenylbiguanide hydrochloride	RS 56812 hydrochloride	RS 67506 hydrochloride	Spiperone hydrochloride	N-Desmethylclozapine	RS 16566 dihydrochloride	Nisoxetine hydrochloride	CP 93129 dihydrochloride	4-P-PDOT	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	8-M-PDOT	ZM 241385	GR 55562 dihydrochloride	WIN 64338 hydrochloride	BW 723C86 hydrochloride	(S)-(-)-Pindolol	2-Cl-IB-MECA	ACPT-II	AM 281	(S)-(+)-Niguldipine hydrochloride	Empty
b	Empty	Galanin (1-30) (human)	PACAP 1-38	SR 57227 hydrochloride	SC 19220	MRS 1220	DH 97	SB 224289 hydrochloride	SB 216641 hydrochloride	SDZ SER 082 fumarate	Abn-CBD	Empty
c	Empty	CP 94253 hydrochloride	GR 113808	Arvanil	VUF 5574	PD 81723	Sphingosine-1-phosphate	SB 204741	SB 228357	SB 221284	L-152,804	Empty
d	Empty	NAS-181	MAFP	BMY 45778	N-Arachidonylglycine	Ghrelin (human)	GR 127935 hydrochloride	Oleylethanolamide	GR 231118	LY 215840	HEMADO	Empty
e	Empty	MRS 1706	SCH 79797 dihydrochloride	Mesulergine hydrochloride	GR 125487 sulfamate	SB 206553 hydrochloride	PIT	L-655,240	CGS 15943	BIIE 0246	N6-Cyclopentyladenosine	Empty
f	Empty	2-Chloro-N6-cyclopentyladenosine	CV 1808	R-96544 hydrochloride	Acifran	NNC 63-0532	Zacopride hydrochloride	WAY 161503 hydrochloride	SR 2640 hydrochloride	Altanserin hydrochloride	Palmitoylisopropylamide	Empty
g	Empty	Seglitide	Ro 60-0175 fumarate	Alytesin	U 46619	[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P	Ritanserin	GR 79236	SB 258585 hydrochloride	AS 19	L-803,087 trifluoroacetate	Empty
h	Empty	L-817,818	PNU 142633	PSB 1115	PSB 10 hydrochloride	PSB 11 hydrochloride	PSB 36	Cinalukast	SDZ 205-557 hydrochloride	Iloprost	Exendin-3 (9-39) amide	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	RS 102895 hydrochloride	NTNCB hydrochloride	WAY 629 hydrochloride	CGP 71683 hydrochloride	PD 160170	PNU 22394 hydrochloride	LY 255283	[Des-octanoyl]-Ghrelin (human)	L-692,585	SCH 58261	Empty
b	Empty	FPL 55712	2'-MeCCPA	SEW 2871	O-1918	Prostaglandin E2	Leukotriene B4	SR 142948	SR 49059	MK 571	WEB 2086	Empty
c	Empty	CGH 2466 dihydrochloride	EMD 386088 hydrochloride	LY 320135	JTE 013	L-371,257	BIBO 3304 trifluoroacetate	[Pyr1]-Apelin-13	NNC 26-9100	(1R,1'S,3'R/1R,1'R,3'S)-L-054,264	SCH 442416	Empty
d	Empty	SDZ WAG 994	IBC 293	JTE 907	(±)-AC 7954 hydrochloride	Melperone hydrochloride	MRS 2693 trisodium salt	Trap 101	APC 366	L-161,982	T 98475	Empty
e	Empty	LP 44	Tocrifluor T1117	SUN-B 8155	PNU 109291	ZK 756326	Melanotan II	α-MSH	TCB-2	J 113863	(±)-J 113397	Empty
f	Empty	PD 176252	RWJ 56110	L-703,664 succinate	L-368,899 hydrochloride	Fananserin	Bucindolol	BIBP 3226 trifluoroacetate	PSB 0474	AG 045572	MRS 1754	Empty
g	Empty	Nefazodone hydrochloride	O-1602	Alprenolol hydrochloride	Arachidonyl serotonin	Ro 04-6790	MRS 2690	LP 12 hydrochloride	PAF (C16)	(R)-(+)-m-Nitrobiphenyline oxalate	DSP-4	Empty
h	Empty	Epoprostenol	1-Methylpsilocin	THIQ	Sulprostone	Desipramine hydrochloride	LY 272015 hydrochloride	LY 334370 hydrochloride	CJ 033466	NBI 35965 hydrochloride	UDP disodium salt	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	BMS CCR2 22	2-Chloroadenosine	BAY-u 9773	Talopram hydrochloride	SB 699551	SB 399885 hydrochloride	PSB 603	PSB 0788	alpha,beta-Methyleneadenosine 5'-triphosphate trisodium salt	PACAP 6-38	Empty
b	Empty	SCH 221510	BMS 193885	UTPγS trisodium salt	2-ThioUTP tetrasodium salt	NPS ALX Compound 4a dihydrochloride	Oxprenolol hydrochloride	8-(3-Chlorostyryl)caffeine	BGC 20-761	L-798,106	SLV 320	Empty
c	Empty	ATC 0175 hydrochloride	SNAP 94847 hydrochloride	LY 393558	NS 304	PSN 375963 hydrochloride	ATC 0065	M40	S 25585	Cyclosomatostatin	ML 10302 hydrochloride	Empty
d	Empty	LU AA33810	SB 657510	SB 612111 hydrochloride	(±)-5'-Chloro-5'-deoxy-ENBA	Org 12962 hydrochloride	CYM 5442 hydrochloride	W146	FR 171113	Donitriptan hydrochloride	PF 514273	Empty
e	Empty	NPY 5RA972	SGS 518 oxalate	SR 48692	SC 51089	CP 135807	R 568 hydrochloride	NF 340	MRS 2768 tetrasodium salt	WAY 207024 dihydrochloride	NF 546	Empty
f	Empty	SF 11	WAY 208466 dihydrochloride	NIDA 41020	OPC 21268	WAY 267464 dihydrochloride	ANR 94	YIL 781	NPEC-caged-noradrenalin	NPEC-caged-serotonin	Zotepine	Empty
g	Empty	16,16-Dimethyl Prostaglandin E2	BMS 470539 dihydrochloride	MJ 15	TCS 2510	PF9 tetrasodium salt	LY 266097 hydrochloride	ML 145	MDL 100907	AS 1269574	VPC 23019	Empty
h	Empty	EMDT oxalate	Prostaglandin F2α	XCC	GW 803430	TC-O 9311	[D-Trp8]-γ-MSH	RP 001 hydrochloride	CID 2745687	Pamoic acid disodium salt	TC 14012	Empty

	1	2	3	4	5	6	7	8	9	10	11	12
a	Empty	SB 268262	FC 131	ST 1936 oxalate	Talsupram hydrochloride	Bicifadine hydrochloride	TC-SP 14	BIMU 8	Calhex 231 hydrochloride	(+)-Fluprostenol	3,5-DHBA	Empty
b	Empty	(±)-SLV 319	Tegaserod maleate	TC OT 39	N,N-Dimethylsphingosine	GW 627368	Strontium chloride	Lu AA 47070	MA 2029	DR 4485 hydrochloride	TC-G 1000	Empty
c	Empty	GSK 1562590 hydrochloride	Prosaptide TX14(A)	ML 154	NBOH-2C-CN hydrochloride	TCS 3035	NIBR189	Pimavanserin	MK-571 sodium salt hydrate	Scopine	Silodosin	Empty
d	Empty	Fingolimod hydrochloride	Adrenaline	Hydrocortisone	Corticosterone	Phloretin	Grifolic acid	Empty	Empty	Empty	Empty	Empty
e	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty
f	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty
g	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty
h	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty	Empty

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Description & Advantages

Storage and Shipping Information

Contents of GPCR/G protein Compound Library

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