Products with
Inhibitors bioactivity
Cat.No.
|
Product Name
|
BCN4014 |
Methyl 4-hydroxycinnamate
|
Methyl 4-hydroxycinnamate is a model chromophore of the Photoactive Yellow Protein (PYP). Methyl 4-hydroxycinnamate can reduce IL-8 secretion at 10 ug/mL treatment concentrations; it may significantly contribute to antibacterial activities of Noni leaves. |
BCN4023 |
Methyl ferulate
|
1. Methyl ferulate is a possible inhibitor of the mitogen activated phosphor kinase pathway.
2. Methyl ferulate could be a potential anti-inflammatory agent isolated for the first time in medicinal plant S. tuberosa.
3. Methyl ferulate has promising anthelmintic activity against Haemonchus contortus. |
BCN4040 |
Nagilactone C
|
1. Nagilactone C possesses potent antiproliferative activity against human fibrosarcoma and murine colon carcinoma tumor cell lines exhibiting ED50 values of 2.3 and 1.2 microg/ml, respectively.
2. Nagilactone C and phyllanthoside are novel protein synthesis inhibitors, they are specific for the eukaryotic translation apparatus, function in vivo and in vitro, and interfere with translation elongation.
3. Nagilactone C shows high insecticidal activity against second-instar nymphs of Eocanthecona furcellata. |
BCN4046 |
Thevetin B
|
1. Thevetin B is a cardiac glycoside.
2. Thevetin A and thevetin B are Na+-, K+-dependent adenosinetriphosphatase (Na+,K+-ATPase) (EC 3.6.1.3) inhibitors. |
BCN4048 |
N-Nornuciferine
|
1. N-Nornuciferine can competitively inhibit CYP2D6 activity with Ki values of 2.34 uM. |