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Products for Muscarinic Receptor

  1. Cat.No. Product Name Information
  2. BCC6939 AF-DX 116 Otenzepad (AF-DX 116) is a selective and competitive M2 muscarinic acetylcholine receptor antagonist, with IC50 values of 640 nM and 386 nM for rabbit peripheral lung and rat heart, respectively. AF-DX 116
  3. BCC1470 Cevimeline Cevimeline (AF-102B) is a quinuclidine derivative of acetylcholine and a selective and orally active muscarinic M1 and M3 receptor agonist. Cevimeline stimulates secretion by the salivary glands and can be used as a sialogogue for xerostomia. Cevimeline can cross the blood-brain barrier (BBB). Cevimeline
  4. BCC7907 VU 0357017 hydrochloride VU0357017 hydrochloride is a highly selective M1 agonists that appear to act at an allosteric site to activate the receptor (EC50 = 477 ± 172 nM; pEC50 = 6.37 ± 0.15). VU 0357017 hydrochloride
  5. BCC7766 VU 0255035 VU 0255035
  6. BCC7729 VU 0238429 VU 0238429 is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5), with an EC50 of 1.16 μM. VU 0238429
  7. BCC7024 AF-DX 384 AF-DX 384
  8. BCC6627 Arecaidine but-2-ynyl ester tosylate Arecaidine but-2-ynyl ester tosylate
  9. BCC6707 5-Methylfurmethiodide 5-Methylfurmethiodide
  10. BCC6164 VU 0365114 VU 0365114 is a mAChR M5 positive allosteric modulator, with an EC50 of 2.7 μM. VU 0365114
  11. BCC4565 Biperiden HCl Biperiden Hydrochloride (KL 373 Hydrochloride) is an antiparkinsonian agent, which is the selective central M1 cholinoreceptors blocker. Biperiden HCl
  12. BCC7314 AQ-RA 741 Selective, high affinity M<sub>2</sub> antagonist AQ-RA 741
  13. BCC4586 Tolterodine tartrate Tolterodine Tartrate (Kabi-2234; PNU-200583E) is a potent muscarinic receptor antagonist and shows selectivity for the urinary bladder over salivary glands in vivo. Tolterodine tartrate
  14. BCC7418 Zamifenacin fumarate Zamifenacin fumarate (UK-76654 fumarate) is a potent gut-selective muscarinic M3 receptor antagonist. Zamifenacin significantly reduces colonic motility in irritable bowel syndrome. Zamifenacin fumarate
  15. BCC7263 DAU 5884 hydrochloride DAU 5884 hydrochloride
  16. BCC1516 Darifenacin Darifenacin(UK88525) is a selective M3 muscarinic receptor antagonist with pKi of 8.9. Darifenacin
  17. BCC4567 Darifenacin HBr Darifenacin hydrobromide (UK-88525 hydrobromide) is a selective M3 muscarinic receptor antagonist with pKi of 8.9. Darifenacin HBr
  18. BCC7061 (S)-(+)-Dimethindene maleate (S)-(+)-Dimethindene maleate
  19. BCC7427 Milameline hydrochloride Milameline hydrochloride
  20. BCC6628 Arecaidine propargyl ester tosylate Arecaidine propargyl ester tosylate
  21. BCC6946 Telenzepine dihydrochloride Telenzepine dihydrochloride
  22. BCC1471 Cevimeline hydrochloride hemihydrate Cevimeline hydrochloride hemihydrate (SNI-2011) is a quinuclidine derivative of acetylcholine and a selective and orally active muscarinic M1 and M3 receptor agonist. Cevimeline hydrochloride hemihydrate stimulates secretion by the salivary glands and can be used as a sialogogue for xerostomia. Cevimeline hydrochloride hemihydrate can cross the blood-brain barrier (BBB). Cevimeline hydrochloride hemihydrate
  23. BCC6814 Oxotremorine sesquifumarate Oxotremorine sesquifumarate
  24. BCC6661 4-DAMP 4-DAMP
  25. BCC6217 PTAC oxalate PTAC oxalate
  26. BCC4583 5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM) Desfesoterodine (PNU-200577; Desfesoterodine) is a potent and selective muscarinic receptor antagonist with a Kb and a pA2 of 0.84 nM and 9.14, respectively. 5-hydroxymethyl Tolterodine (PNU 200577, 5-HMT, 5-HM)
  27. BCC6682 W-84 dibromide W-84 dibromide
  28. BCC7145 PD 102807 PD 102807
  29. BCC4580 Solifenacin succinate Solifenacin Succinate (YM905) is a novel muscarinic receptor antagonist with pKis of 7.6, 6.9 and 8.0 for M1, M2 and M3 receptors, respectively. Solifenacin succinate
  30. BCC7556 (+)-Muscarine iodide (+)-Muscarine iodide
  31. BCC7389 J 104129 fumarate J 104129 fumarate
  32. BCC4584 Fesoterodine Fumarate Fesoterodine Fumarate is an antimuscarinic agent and is rapidly de-esterified to its active metabolite 5-hydroxymethyl tolterodine that is a muscarinic receptor antagonist. Fesoterodine Fumarate
  33. BCC6923 Pirenzepine dihydrochloride Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist. Pirenzepine dihydrochloride
  34. BCC4575 Aclidinium Bromide Aclidinium Bromide(LAS 34273; LAS-W 330) is a long-acting, inhaled muscarinic antagonist as a maintenance treatment for chronic obstructive pulmonary disease (COPD). Aclidinium Bromide
  35. BCC6920 Oxotremorine M Oxotremorine M iodide is a potent and non-selective muscarinic acetylcholine receptor (mAChR) agonist. Oxotremorine M iodide potentiates NMDA receptors by muscarinic receptor dependent and independent mechanisms. Oxotremorine M
  36. BCC7042 McN-A 343 McN-A 343
  37. BCC7577 VU 10010 VU 10010
  38. BCC2022 Umeclidinium bromide Umeclidinium bromide is a novel mAChR antagonist. The affinity (Ki) of Umeclidinium bromide for the cloned human M1-M5 mAChRs ranges from 0.05 to 0.16 nM. Umeclidinium bromide
  39. BCC6655 Nitrocaramiphen hydrochloride Nitrocaramiphen hydrochloride

Items 1 to 38 of 38 total

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