Hot Natural Products & Bioactive Compounds
BioCrick offers high-purity natural products and bioactive compounds for scientific research. Our natural product collection includes compounds derived from plants, microorganisms and other biological sources and is widely used in pharmacological, biochemical and drug discovery research.
Natural products remain an important source of bioactive molecules and drug leads. BioCrick provides researchers with high-quality natural product compounds together with catalog numbers, product information and biological activity data.
Hot Products from BioCrick
Showing 825 - 832 of 9359 hot products
| Catalog No. | Product Name |
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| BCC4343 | Betaxolol HCl |
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Selective <span class='symbol'>β</span><sub>1</sub>-adrenoceptor antagonist.
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| BCC4344 | Bisoprolol fumarate |
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A selective <span class='symbol'>β</span><sub>1</sub>-adrenergic antagonist. Has a K<sub>d</sub> of 2-3 nM at the <span class='symbol'>β</span><sub>1</sub> receptor and a <span class='symbol'>β</span><sub>1</sub>/<span class='symbol'>β</span><sub>2</sub> selectivity of approximately 100-fold.
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| BCC4347 | Dexmedetomidine HCl |
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Active isomer of medetomidine, a potent, highly selective <span class='symbol'>α</span><sub>2</sub>-adrenoceptor agonist (K<sub>i</sub> values are 1.08 and 1750 nM for <span class='symbol'>α</span><sub>2</sub>- and <span class='symbol'>α</span><sub>1</sub>-adrenoceptors respectively). Displays greater selectivity over <span class='symbol'>α</span><sub>1</sub>-adrenoceptors than clonidine and UK 14,304 (1620-, 220- and 300-fold respectively). Active <em>in vivo</em>; displays hypotensive, bradycardic, sedative, anxiolytic, hypothermic and analgesic effects.
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| BCC4349 | Formoterol Hemifumarate |
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Potent, selective and long-acting <span class='symbol'>β</span><sub>2</sub>-adrenoceptor agonist. Displays 330-fold selectivity for <span class='symbol'>β</span><sub>2</sub> over <span class='symbol'>β</span><sub>1</sub> receptors (pK<sub>d</sub> values are 8.12 and 5.58 respectively). Potently relaxes guinea pig trachea (pD<sub>2</sub> = 9.29), and is longer-acting and 100-fold more potent than salbutamol.
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| BCC4350 | Ivabradine HCl |
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HCN channel blocker (IC50 is approximately 0.5 - 2.5 μM). Bradycardic agent that inhibits If pacemaker current in sinoatrial node cells.
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| BCC4351 | Medetomidine HCl |
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Potent, highly selective <span class='symbol'>α</span><sub>2</sub>-adrenoceptor agonist (K<sub>i</sub> values are 1.08 and 1750 nM for <span class='symbol'>α</span><sub>2</sub>- and <span class='symbol'>α</span><sub>1</sub>-adrenoceptors respectively). Displays greater selectivity over <span class='symbol'>α</span><sub>1</sub>-adrenoceptors than clonidine and UK 14,304 (1620-, 220- and 300-fold respectively). Inhibits twitch response in electrically stimulated mouse vas deferens (pD<sub>2</sub> = 9.0). Active <em>in vivo</em>; displays hypotensive, bradycardic, sedative, anxiolytic, hypothermic and analgesic effects.
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| BCC4353 | Phentolamine Mesylate |
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Non-selective adrenergic α receptor antagonist (pKB = 8.07). Intravenous injection causes hypotension and tachycardia in rats. Intraperitoneal injection in mice increases plasma FGF21 levels.
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| BCC4357 | Tizanidine HCl |
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<span class='symbol'>α</span><sub>2</sub>-adrenergic receptor agonist. Antinociceptive upon epidural administration in rats (IC<sub>50</sub> = 48 nM). Also binds to imidazoline receptor.
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