Hot Natural Products & Bioactive Compounds
BioCrick offers high-purity natural products and bioactive compounds for scientific research. Our natural product collection includes compounds derived from plants, microorganisms and other biological sources and is widely used in pharmacological, biochemical and drug discovery research.
Natural products remain an important source of bioactive molecules and drug leads. BioCrick provides researchers with high-quality natural product compounds together with catalog numbers, product information and biological activity data.
Hot Products from BioCrick
Showing 1705 - 1712 of 9359 hot products
| Catalog No. | Product Name |
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| BCC6107 | Flunitrazepam |
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Ligand at the GABAA receptor benzodiazepine modulatory site. Exhibits hypnotic effects; also displays anxiolytic and sedative properties.
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| BCC6108 | 8-Aminoadenine |
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Adenine receptor agonist (K<sub>i</sub> = 0.0341 <span class='symbol'>μ</span>M in HEK293 cells expressing an adenine binding site). Displays 190-fold increased potency at the human binding site over the rat adenine receptor (rAde1R) (K<sub>i</sub> = 6.51 <span class='symbol'>μ</span>M).
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| BCC6109 | LY 78335 |
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High affinity inhibitor of phenylethanolamine-<em>N</em>-methyltransferase (PNMT) (K<sub>i</sub> = 0.09 <span class='symbol'>μ</span>M <em>in vitro</em>). Suppresses the release of growth hormone in an <em>in vivo</em> rat model.
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| BCC6110 | Fluorobexarotene |
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RXR agonist (K<sub>i</sub> = 12 nM; EC<sub>50</sub> = 43 nM at RXR<span class='symbol'>α</span> receptors). Displays similar RAR agonist activity to bexarotene; exhibits an apparent RXR binding affinity 75% greater than bexarotene.
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| BCC6111 | TCN 237 dihydrochloride |
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Highly potent NR2B-selective NMDA receptor antagonist (K<sub>i</sub> = 0.8 nM); blocks NR2B-mediated calcium influx in Ltk cells (K<sub>i</sub> = 9.7 nM). Selective for NR2B subunit over <span class='symbol'>α</span><sub>1</sub>-adrenergic receptors and hERG channels (IC<sub>50</sub> values are 730 nM and 2900 nM respectively). Displays efficacy in the rat carrageenan-induced mechanical hyperalgesia assay.
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| BCC6112 | 3F8 |
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Potent and selective GSK-3<span class='symbol'>β</span> inhibitor (IC<sub>50</sub> values are 34 and 304 nM in the presence of 10 and 100 <span class='symbol'>μ</span>M ATP respectively).
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| BCC6113 | LPYFD-NH2 |
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Neuroprotective peptide that binds to amyloid beta (A<span class='symbol'>β</span>). Protects neurons against toxic effects of A<span class='symbol'>β</span> (1-42) <em>in vitro</em> and <em>in vivo</em>. Potential therapeutic in the treatment of Alzheimer's Disease.
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| BCC6114 | MM-22 |
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Biotinylated anandamide analog; acts as a probe for visualizing the accumulation and intracellular trafficking of anandamide. Blocks anandamide uptake (IC<sub>50</sub> = 0.5 <span class='symbol'>μ</span>M in HaCaT cells); prevents interaction with FAAH, CB<sub>1</sub> and TRPV1.
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