6'-IodoresiniferatoxinHigh affinity TRPV1 agonist/partial agonist CAS# 335151-55-8 |
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Quality Control & MSDS
3D structure
Package In Stock
Number of papers citing our products
| Cas No. | 335151-55-8 | SDF | Download SDF |
| PubChem ID | 73993817 | Appearance | Powder |
| Formula | C37H39IO9 | M.Wt | 754.6 |
| Type of Compound | N/A | Storage | Desiccate at -20°C |
| Synonyms | 6'-IRTX | ||
| Solubility | Soluble in DMSO > 10 mM | ||
| SMILES | CC1CC2(C3C4C1(C5C=C(C(=O)C5(CC(=C4)COC(=O)CC6=CC(=C(C=C6I)O)OC)O)C)OC(O3)(O2)CC7=CC=CC=C7)C(=C)C | ||
| Standard InChIKey | IITCVPTZKLXSKQ-UHFFFAOYSA-N | ||
| Standard InChI | InChI=1S/C37H39IO9/c1-20(2)35-16-22(4)37-26(33(35)45-36(46-35,47-37)18-23-9-7-6-8-10-23)12-24(17-34(42)30(37)11-21(3)32(34)41)19-44-31(40)14-25-13-29(43-5)28(39)15-27(25)38/h6-13,15,22,26,30,33,39,42H,1,14,16-19H2,2-5H3 | ||
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months. We recommend that you prepare and use the solution on the same day. However, if the test schedule requires, the stock solutions can be prepared in advance, and the stock solution must be sealed and stored below -20℃. In general, the stock solution can be kept for several months. Before use, we recommend that you leave the vial at room temperature for at least an hour before opening it. |
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| About Packaging | 1. The packaging of the product may be reversed during transportation, cause the high purity compounds to adhere to the neck or cap of the vial.Take the vail out of its packaging and shake gently until the compounds fall to the bottom of the vial. 2. For liquid products, please centrifuge at 500xg to gather the liquid to the bottom of the vial. 3. Try to avoid loss or contamination during the experiment. |
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| Shipping Condition | Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other couriers with RT, or blue ice upon request. | ||
| Description | High affinity TRPV1 (VR1) vanilloid receptor partial agonist (Ki = 0.71 nM; EC50 = 130 nM at human VR1). Displays partial agonism at human VR1 and full agonism at rat VR1. |
6'-Iodoresiniferatoxin Dilution Calculator
6'-Iodoresiniferatoxin Molarity Calculator
| 1 mg | 5 mg | 10 mg | 20 mg | 25 mg | |
| 1 mM | 1.3252 mL | 6.626 mL | 13.2521 mL | 26.5041 mL | 33.1301 mL |
| 5 mM | 0.265 mL | 1.3252 mL | 2.6504 mL | 5.3008 mL | 6.626 mL |
| 10 mM | 0.1325 mL | 0.6626 mL | 1.3252 mL | 2.6504 mL | 3.313 mL |
| 50 mM | 0.0265 mL | 0.1325 mL | 0.265 mL | 0.5301 mL | 0.6626 mL |
| 100 mM | 0.0133 mL | 0.0663 mL | 0.1325 mL | 0.265 mL | 0.3313 mL |
| * Note: If you are in the process of experiment, it's necessary to make the dilution ratios of the samples. The dilution data above is only for reference. Normally, it's can get a better solubility within lower of Concentrations. | |||||
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Synthesis and in vitro evaluation of a novel iodinated resiniferatoxin derivative that is an agonist at the human vanilloid VR1 receptor.[Pubmed:11934585]
Bioorg Med Chem Lett. 2002 Apr 22;12(8):1189-92.
Using a 'directed' iodination procedure, novel iodo-resiniferatoxin congeners were synthesized from 4-acetoxy-3-methoxyphenylacetic acid and resiniferinol- 9,13,14-ortho-phenylacetate (ROPA). The 2-iodo-4-hydroxy-5-methoxyphenylacetic acid ester of resiniferinol 5 displayed high affinity binding (K(i)=0.71 nM) for the human vanilloid VR1 receptor and functioned as a partial agonist.
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