Hot Natural Products & Bioactive Compounds
BioCrick offers high-purity natural products and bioactive compounds for scientific research. Our natural product collection includes compounds derived from plants, microorganisms and other biological sources and is widely used in pharmacological, biochemical and drug discovery research.
Natural products remain an important source of bioactive molecules and drug leads. BioCrick provides researchers with high-quality natural product compounds together with catalog numbers, product information and biological activity data.
Hot Products from BioCrick
Showing 2465 - 2472 of 9359 hot products
| Catalog No. | Product Name |
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| BCC7023 | L-655,708 |
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Potent, selective inverse agonist for the benzodiazepine site of GABAA receptors containing the α5 subunit (Ki = 0.45 nM). Displays 50-100-fold selectivity over GABAA receptors containing α1, α2, α3 or α6 subunits in combination with β3 and γ2. Enhances LTP in a mouse hippocampal slice model and increases spatial learning, without displaying proconvulsant activity.
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| BCC7024 | AF-DX 384 |
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Potent M2/M4 selective antagonist (pKi values are 8.22, 8.00, 7.51, 7.18 and 6.27 at human M2, M4, M1, M3 and M5 receptors respectively).
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| BCC7025 | Nafadotride |
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Highly potent, competitive, preferential dopamine D<sub>3</sub> receptor antagonist. K<sub>i</sub> values are 0.52, 5, and 269 nM for human cloned D<sub>3</sub>, D<sub>2</sub> and D<sub>4</sub> receptors respectively. Centrally active upon systemic administration.
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| BCC7026 | Arvanil |
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Cannabinoid CB<sub>1</sub> and vanilloid TRPV1 (VR1) agonist (K<sub>i</sub> values are 0.5 and 0.3 <span class='symbol'>μ</span>M respectively). Also inhibits the anandamide transporter (IC<sub>50</sub> = 3.6 <span class='symbol'>μ</span>M). Analgesic, vasodilatory and anti-inflammatory <em>in vivo</em>.
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| BCC7027 | P1075 |
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Potent K<sub>ir</sub>6 (K<sub>ATP</sub>) channel opener (EC<sub>50</sub> for relaxation of rat aorta = 7.5 nM). Binds to SUR2A and SUR2B with high affinity (K<sub>d</sub> values are 17 and 3 nM respectively).
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| BCC7028 | MG 624 |
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A selective antagonist for neuronal <span class='symbol'>α</span>7 subunit- containing nAChR subtypes. Inhibits <span class='symbol'>α</span>-Bgtx binding to chick <span class='symbol'>α</span>7 and <span class='symbol'>α</span>4<span class='symbol'>β</span>2 subtypes with K<sub>i</sub> values of 106 nM and 84 <span class='symbol'>μ</span>M respectively.
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| BCC7029 | U 99194 maleate |
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Potent, selective D<sub>3</sub> antagonist. K<sub>i</sub> values are 160, 2281 and > 10000 nM for human cloned D<sub>3</sub>, D<sub>2</sub> and D<sub>4</sub> receptors respectively.
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| BCC7030 | VUF 5574 |
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Potent, selective, competitive antagonist for the human adenosine A3 receptor (Ki = 4 nM). Displays ≥ 2500-fold selectivity over A1 and A2A receptors.
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