Hot Natural Products & Bioactive Compounds
BioCrick offers high-purity natural products and bioactive compounds for scientific research. Our natural product collection includes compounds derived from plants, microorganisms and other biological sources and is widely used in pharmacological, biochemical and drug discovery research.
Natural products remain an important source of bioactive molecules and drug leads. BioCrick provides researchers with high-quality natural product compounds together with catalog numbers, product information and biological activity data.
Hot Products from BioCrick
Showing 2481 - 2488 of 9359 hot products
| Catalog No. | Product Name |
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| BCC7039 | Levcromakalim |
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Active enantiomer of the prototypical K<sub>ir</sub>6 (K<sub>ATP</sub>) channel opener cromakalim. Hypotensive and airways relaxant. IC<sub>50</sub> = 490 nM in guinea pig trachea.
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| BCC7040 | SB 221284 |
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Potent, selective 5-HT2C/2B receptor antagonist. pKi values are 6.4, 7.9 and 8.6 for 5-HT2A, 2B and 2C receptors respectively. Centrally active upon systemic administration in vivo.
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| BCC7041 | L-152,804 |
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Potent, selective non-peptide neuropeptide Y Y5 receptor antagonist (Ki = 26 nM for hY5). Displays > 300-fold selectivity over hY1, hY2, and hY4 receptors. Causes weight loss in diet-induced obese mice by modulating food intake and energy expenditure. Centrally active upon oral administration in vivo.
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| BCC7042 | McN-A 343 |
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Selective muscarinic M1 receptor agonist. Selectivity for M1 over other muscarinic receptor types appears to arise from a high efficacy at M1 receptors.
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| BCC7043 | NF 449 |
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Potent purinergic receptor antagonist that displays high selectivity for P2X<sub>1</sub> (IC<sub>50</sub> values are 0.28, 0.69, 120, 1820, 47000 and > 300000 nM for rP2X<sub>1</sub>, rP2X<sub>1+5</sub>, rP2X<sub>2+3</sub>, rP2X<sub>3</sub>, rP2X<sub>2</sub> and P2X<sub>4</sub> receptors respectively). Provides antithrombotic protection <em>in vivo</em>. Also acts as a G<sub>s<span class='symbol'>α</span></sub>-selective antagonist.
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| BCC7044 | VDM 11 |
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A potent and selective inhibitor of the anandamide membrane transporter (AMT) with IC<sub>50</sub> values of 4-11 <span class='symbol'>μ</span>M. Displays negligible agonist activity at the hVR1 receptor and very weak action at CB<sub>1</sub> and CB<sub>2</sub> receptors. K<sub>i</sub> values are > 5-10 <span class='symbol'>μ</span>M at CB<sub>1</sub> and CB<sub>2</sub>. Active <em>in vivo</em>. Also available in water-soluble emulsion.
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| BCC7045 | (RS)-3,4-DCPG |
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Systemically active anticonvulsant that is 30-100-fold more potent <em>in vivo</em> than the separate enantiomers (S)-3,4-DCPG or (R)-3,4,-DCPG.
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| BCC7046 | (R)-3,4-DCPG |
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AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors. (<em>RS</em>)-3,4-DCPG and (<em>S</em>)-3,4-DCPG also available.
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