Hot Natural Products & Bioactive Compounds
BioCrick offers high-purity natural products and bioactive compounds for scientific research. Our natural product collection includes compounds derived from plants, microorganisms and other biological sources and is widely used in pharmacological, biochemical and drug discovery research.
Natural products remain an important source of bioactive molecules and drug leads. BioCrick provides researchers with high-quality natural product compounds together with catalog numbers, product information and biological activity data.
Hot Products from BioCrick
Showing 3225 - 3232 of 9359 hot products
| Catalog No. | Product Name |
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| BCC7795 | SKF 86466 hydrochloride |
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Potent and selective <span class='symbol'>α</span><sub>2</sub> antagonist at pre- and post-junctional <span class='symbol'>α</span><sub>2</sub>-adrenoceptors (K<sub>i</sub> values are 13 and 17 nM respectively). Exhibits antihypertensive activity in a rat model.
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| BCC7796 | (±)-PPCC oxalate |
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Selective sigma (<span class='symbol'>σ</span>) receptor ligand. Displays high affinity for <span class='symbol'>σ</span><sub>1</sub>; also binds at <span class='symbol'>σ</span><sub>2</sub> sites (K<sub>i</sub> = 1.5 nM and 50.8 nM respectively). Selective over a range of receptor types including dopaminergic and muscarinic receptors, DAT and SERT.
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| BCC7797 | BCTC |
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Orally effective vanilloid receptor 1 (TRPV1 receptor) antagonist. Inhibits acid- and capsaicin-induced activation of rat TRPV1 receptors (IC50 values are 6.0 and 35 nM respectively). Displays analgesic properties in rat models of inflammatory and neuropathic pain. CNS penetrant.
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| BCC7798 | TCS 2210 |
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Inducer of neuronal differentiation in mesenchymal stem cells (MSCs) with specific phenotype change. Increases expression of neuronal markers <span class='symbol'>β</span>-III tubulin and NSE without cytotoxicity.
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| BCC7799 | FFN 511 |
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Fluorescent false neurotransmitter (FFN). Targets neuronal vesicular monoamine transporter (VMAT) 2; inhibits serotonin binding to VMAT2 (IC<sub>50</sub> = 1 <span class='symbol'>μ</span>M).
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| BCC7800 | MRS 2768 tetrasodium salt |
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Selective P2Y<sub>2</sub> agonist (EC<sub>50</sub> = 1.89 <span class='symbol'>μ</span>M). Displays no affinity for human P2Y<sub>4</sub> or P2Y<sub>6</sub> receptors.
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| BCC7801 | PG 01037 dihydrochloride |
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Dopamine D<sub>3</sub> receptor antagonist; 133-fold selective for D<sub>3</sub> over D<sub>2</sub> receptors <em>in vitro</em> (K<sub>i</sub> values are 0.70, 93.3 and 375 nM for D<sub>3</sub>, D<sub>2</sub> and D<sub>4</sub> receptors respectively). Attenuates abnormal involuntary movements associated with L-DOPA in rat models of Parkinson's disease. Inhibits the effects of methamphetamine; attenuates drug-induced behaviors <em>in vivo</em>.
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| BCC7802 | WAY 207024 dihydrochloride |
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Gonadotropin releasing hormone receptor (GnRH-R) antagonist. Exhibits potent affinity (IC50 values are 12 and 71 nM for human and rat GnRH receptors respectively). Lowers plasma leuteinizing hormone levels in the rat. Orally active.
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