Endocrinology and Hormones
The endocrine system is an information signaling system that coordinates most bodily functions. It senses environmental changes and secretes corresponding hormones to coordinate metabolism, maintain homeostasis, and regulate growth and development.
Products for Endocrinology and Hormones
- GnRH(4)
- Estrogen/progestogen Receptor(50)
- Opioid Receptor(70)
- RAAS(7)
- Androgen Receptor(24)
- Aromatase(5)
- 5-alpha Reductase(3)
- Thyroid hormone Receptor(1)
- Non-selective AT(2)
- CRTH2(2)
- Cat.No. Product Name Information
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BCC1037
Angiotensin 1/2 + A (2 - 8)
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BCC4366
Spironolactone
Spironolactone is a potent antagonist of the androgen receptor.
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BCC6368
Morphine hydrochloride
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BCN2748
Dimethylcurcumin
Dimethylcurcumin (ASC-J9) is an androgen receptor degradation enhancer that effectively suppresses castration resistant prostate cancer cell proliferation and invasion.
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BCC7939
(R)-DPN
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BCC7903
ERB 041
Prinaberel(ERB-041) is a potent and selective ERbeta agonist; being >200-fold selective for ERbeta.
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BCN2201
Estrone
Estrone is an estrogenic hormone.
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BCN2855
4',7-Isoflavandiol
(-)-(S)-Equol is a high affinity ligand for estrogen receptor β with a Ki of 0.73 nM.
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BCC5215
Buprenorphine hydrochloride
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BCC4491
Erteberel (LY500307)
Erteberel (LY500307) is a potent and selective estrogen receptor beta (ERβ) agonist with Ki and EC50 of 1.54 nM and 3.61 nM, respectively. Anti-tumor activities.
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BCC5230
Etonogestrel
Etonogestrel is a steroidal progestin used in hormonal contraceptives.
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BCC4382
Tamoxifen Citrate
Tamoxifen Citrate (ICI 46474) is a selective estrogen receptor modulator (SERM) which blocks estrogen action in breast cells and can activate estrogen activity in other cells, such as bone, liver, and uterine cells.Tamoxifen Citrate is a potent Hsp90 activator and enhances the Hsp90 molecular chaperone ATPase activity. Tamoxifen Citrate activates autophagy and induces apoptosis.
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BCC6093
Nalmefene - d3
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BCC4369
Formestane
Formestane is a second generation selective aromatase inhibitor with an IC50 of 80 nM.
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BCC6442
Chlorotrianisene
Chlorotrianisene is a long-acting non-steroidal estrogen and an orally active estrogen receptor modulator. Chlorotrianisene exhibits antiestrogenic activity. Chlorotrianisene potently inhibits the enzyme COX-1 and inhibits platelet aggregation in whole blood.
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BCC3777
Ethinyl Estradiol
Ethynyl Estradiol (17α-Ethynylestradiol;Ethynylestradiol) is an orally bio-active estrogen used in almost all modern formulations of combined oral contraceptive pills.
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BCC7497
α-Estradiol
Alpha-Estradiol is a weak estrogen and a 5α-reductase inhibitor which is used as a topical medication in the treatment of androgenic alopecia.
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BCC1035
Angiotensin 1/2 (1-5)
Angiotensin I/II 1-5 is a peptide that contains the amino acids 1-5, which is converted from Angiotensin I/II. Angiotensin I is formed by the action of renin on angiotensinogen. Angiotensin II is produced from angiotensin I. Angiotensin II has been investigated for the treatment, basic science, and diagnostic of Hypertension, Renin Angiotensin System, and Idiopathic Membranous Nephropathy.
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BCC5831
[Leu5]-Enkephalin
[Leu5]-Enkephalin is a pentapeptides with morphine like properties. [Leu5]-Enkephalin is a five amino acid endogenous peptide that acts as an agonist at opioid receptors.
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BCC7857
Nalmefene hydrochloride
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BCC4920
Meptazinol HCl
Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]dihydromorphine binding with IC50 of 58 nM.
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BCC4490
Gestodene
Gestodene(SHB 331;WL 70) is a progestogen hormonal contraceptive.
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BCC1754
MK-0773
MK-0773 is a selective androgen receptor modulators (SARMs) that binds to AR with an IC50 of 6.6 nM.
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BCC2140
Captopril
Captopril (SQ-14534) is a potent, competitive inhibitor of angiotensin-converting enzyme (ACE).
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BCC1425
BMS-564929
BMS-564929 is an androgen receptor (AR) agonist, binds to androgen receptor (AR) with a Ki of 2.11±0.16 nM.
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BCC6064
DADLE
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BCC5352
Goserelin Acetate
Goserelin(ICI 118630) is an injectable gonadotropin releasing hormone superagonist (GnRH agonist).
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BCC1023
Acetyl Angiotensinogen (1-14), porcine
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BCC6665
(±)-U-50488 hydrochloride
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BCC6015
(Z)-4-Hydroxytamoxifen
4-Hydroxytamoxifen is a selective estrogen receptor modulator (SERM).
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BCC4485
Medroxyprogesterone acetate
Medroxyprogesterone acetate is a widely used synthetic steroid by its interaction with progesterone, androgen and glucocorticoid receptors。
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BCC5121
XCT790
XCT-790 is a potent and selective inverse agonist for ERRα with an IC50 value of 0.37 μM. XCT-790 induces cell death in chemotherapeutic resistant cancer cells. XCT-790 (Compound 12) is inactive against ERRγ and the estrogen receptors ERα and ERβ.
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BCC6850
β-Funaltrexamine hydrochloride
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BCC7719
Estropipate
Estropipate is a form of estrogen, used to treat symptoms of menopause, also used to prevent osteoporosis.
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BCC1740
Methylnaltrexone Bromide
Methylnaltrexone (Bromide) is a peripheral-acting opioid receptor antagonist that acts on the gastrointestinal tract to decrease opioid-induced constipation.
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BCC1701
Leuprolide Acetate
Leuprolide acetate (Leuprorelin acetate) is a potent gonadotropin-releasing hormone receptor agonist used for the treatment of prostate cancer, endometriosis, uterine fibroids.
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BCC5718
DSLET
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BCC5255
Oxymorphone
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BCC6979
TCPOBOP
TCPOBOP is a constitutive androstane receptor (CAR) agonist that induces robust hepatocyte proliferation and hepatomegaly without any liver injury or tissue loss. TCPOBOP attenuates Fas-induced murine liver injury by altering Bcl-2 proteins.
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BCC5797
BAM 22P
BAM-22P, a highly potent opioid peptide, is a potent opioid agonist.
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BCC6958
DAMGO
DAMGO is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR.
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BCC1671
JDTic 2HCl
JDTic (dihydrochloride) is a potent antagonist of kappa-opioid receptors (KOR), blocking the κ-agonist U50, 488-induced antinociception.
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BCC1336
Alarelin Acetate
Alarelin acetate is a synthetic GnRH agonist.
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BCC4506
AZD1981
AZD1981 is a potent and selective CRTh2 antagonist; displaces radio-labelled PGD2 from human recombinant DP2 with high potency (pIC50 = 8.4).
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BCC7596
Dynorphin A
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BCC7447
PHTPP
PHTPP is a selective ERβ antagonist.
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BCC4488
Raloxifene HCl
Raloxifene hydrochloride (LY156758 hydrochloride; LY139481 hydrochloride) is a second generation selective and orally active estrogen receptor modulator. Raloxifene hydrochloride produces estrogen-agonistic effects on bone and lipid metabolism and estrogen-antagonistic effects on uterine endometrium and breast tissue.
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BCC5987
Dynorphin B
Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.
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BCC5864
PL 017
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BCC5677
ICI 154,129
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BCC5875
Salvinorin A
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BCC4484
Hexestrol
Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
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BCC7451
Y 134
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BCC4479
Altrenogest
Altrenogest (Allyltrenbolone) is a progestogen structurally related to veterinary steroid trenbolone.
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BCC1265
ADL5859 HCl
ADL5859 is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel.
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BCC3910
TOK-001
Galeterone (TOK-001) is a multifunctional antiandrogen and CYP17 inhibitor (IC50=47 nM) in castration resistant prostate cancer (CRPC).
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BCC7082
FIT
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BCC1467
Cebranopadol
Cebranopadol is an analgesic NOP and opioid receptor agonist with Kis/EC50s of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, 18 nM/110 nM for human NOP, MOP, KOP and delta-opioid peptide (DOP) receptor, respectively.
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BCC6838
BNTX maleate
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BCC5508
NVP-QAV680
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BCC6710
Naloxonazine dihydrochloride
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BCC6045
G-1
G-1 is a nonsteroidal, high-affinity and selective agonist of GPR30 with a Ki of 11 nM.
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BCC5758
DPDPE
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BCC5675
ICI 174,864
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BCC3792
Imidapril HCl
Imidapril hydrochloride (TA-6366) is the hydrochloride salt of Imidapril, an angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.
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BCC2010
Toremifene
Toremifene (NK 622; FC 1157a) is a second-generation selective estrogen-receptor modulator (SERM) in development for the prevention of osteoporosis.
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BCC4487
Toremifene Citrate
Toremifene Citrate(NK 622; FC 1157a) is a second-generation selective estrogen-receptor modulator (SERM) in development for the prevention of osteoporosis.
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BCC2481
Bicalutamide
Bicalutamide is a non-steroidal androgen receptor inhibitor.
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BCC7225
MPP dihydrochloride
MPP dihydrochloride is a highly selective estrogen receptor alpha (ERα) antagonist. MPP dihydrochloride reduces the ratio of p-ERα/ERα.
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BCC1268
MDV3100 (Enzalutamide)
Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells. Enzalutamide is an autophagy activator.
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BCC3724
ARN-509
Apalutamide (ARN-509) is a potent and competitive androgen receptor (AR) antagonist, binding AR with an IC50 of 16 nM.
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BCC4482
Estradiol valerate
Estradiol valerianate (β-estradiol 17-valerate) is a synthetic estrogen widely used in combination with other steroid hormones in hormone replacement therapy drugs.
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BCC2491
Finasteride
Finasteride is an orally active testosterone 5-alpha-reductase inhibitor (Ki= 10 nM).
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BCC6000
Fentanyl citrate