Products for Opioid Receptor

  1. Cat.No. Product Name Information
  2. BCC5780 CTOP CTOP
  3. BCC5776 CTAP CTAP
  4. BCC6773 Naltrindole hydrochloride Naltrindole hydrochloride is a highly potent and selective non-peptide δ opioid receptor antagonist with a Ki of 0.02 nM. Naltrindole hydrochloride
  5. BCC6751 BRL 52537 hydrochloride BRL 52537 hydrochloride
  6. BCC6668 U-54494A hydrochloride U-54494A hydrochloride
  7. BCC6614 nor-Binaltorphimine dihydrochloride Norbinaltorphimine dihydrochloride is a potent and selective κ opioid receptor antagonist. nor-Binaltorphimine dihydrochloride
  8. BCC6666 (-)-U-50488 hydrochloride (-)-U-50488 hydrochloride
  9. BCC6656 (+)-U-50488 hydrochloride (+)-U-50488 hydrochloride
  10. BCC6792 ICI 199,441 hydrochloride ICI 199,441 hydrochloride
  11. BCC5684 Clocinnamox mesylate Clocinnamox mesylate
  12. BCC7425 Cyprodime hydrochloride Cyprodime hydrochloride
  13. BCC5757 Naloxone benzoylhydrazone Naloxone benzoylhydrazone (NalBzoH) is a mixed agonist/antagonist. Naloxone benzoylhydrazone is a prototypic κ3-opioid receptor agonist, and a partial agonist at the cloned μ and δ opioid receptors, and an antagonist at opioid-like NOP receptors. Naloxone benzoylhydrazone has potently analgesia effect. Naloxone benzoylhydrazone
  14. BCC6782 N-Benzylnaltrindole hydrochloride N-Benzylnaltrindole hydrochloride
  15. BCC6806 ICI 204,448 hydrochloride ICI 204,448 hydrochloride
  16. BCC5687 SB 205607 dihydrobromide SB 205607 dihydrobromide
  17. BCC5683 Naltriben mesylate Naltriben mesylate
  18. BCC6233 Deltorphin I Deltorphin I is a δ-opioid receptor agonist with high affinity and selectivity. Deltorphin I
  19. BCC5723 [D-Ala2]-Deltorphin II Deltorphin 2 is a selective peptide agonist for the δ opioid receptor. [D-Ala2]-Deltorphin II
  20. BCC6090 Oxycodone hydrochloride Oxycodone hydrochloride
  21. BCC7083 GR 89696 fumarate GR 89696 fumarate
  22. BCC1719 LY2795050 LY2795050 is a novel selective κ-opioid Receptor (KOR) antagonist (IC50=0.72 nM) and has the potential as a PET tracer to image KOR in vivo. LY2795050
  23. BCC6308 ML 190 ML 190
  24. BCC1349 Alvimopan monohydrate Alvimopan monohydrate (ADL 8-2698 monohydrate) is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. Alvimopan monohydrate
  25. BCC5697 Endomorphin-2 Endomorphin 2, a high affinity, highly selective agonist of the μ-opioid receptor, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. Endomorphin-2
  26. BCC5954 Diprenorphine Diprenorphine
  27. BCC6799 DIPPA hydrochloride DIPPA hydrochloride
  28. BCC5798 BW 373U86 BW 373U86
  29. BCC1347 Alvimopan Alvimopan(LY 246736; ADL 8-2698) is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. Alvimopan
  30. BCC6785 SNC 80 SNC80 (NIH 10815) is a potent, highly selective and non-peptide δ-opioid receptor agonist with a Ki of 1.78 nM and an IC50 of 2.73 nM. SNC80 also selectively activates μ-δ heteromer in HEK293 cells with an EC50 of 52.8 nM. SNC80 shows antinociceptive, antihyperalgesic and antidepressant‐like effects. SNC80 has the potential for multiple headache disorders treatment. SNC 80
  31. BCC1783 Naltrexone Naltrexone
  32. BCC4613 Naltrexone HCl Broad spectrum opioid antagonist,Naltrexone HCl is an opioid receptor antagonist used primarily in the management of alcohol dependence and opioid dependence. Naltrexone HCl
  33. BCC1348 Alvimopan dihydrate Alvimopan dihydrate (ADL 8-2698 dihydrate) is a peripherally acting mu-opioid receptor (PAM-OR, IC50= 1.7 nM) antagonist for accelerating gastrointestinal recovery after surgery. Alvimopan dihydrate
  34. BCC7103 SNC 162 SNC 162
  35. BCC5672 N-MPPP Hydrochloride N-MPPP Hydrochloride
  36. BCC6143 AR-M 1000390 hydrochloride AR-M 1000390 hydrochloride is an exceptionally selective, potent δ opioid receptor agonist with an EC50 of 7.2±0.9 nM for δ agonist potency. AR-M 1000390 hydrochloride
  37. BCC3800 JTC-801 JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist, binding to ORL1 receptor with a Ki value of 8.2 nM. JTC-801
  38. BCC7054 SDM25N hydrochloride SDM25N hydrochloride
  39. BCC4380 Loperamide HCl Loperamide (hydrochloride) (R-18553 (hydrochloride)) is an opioid receptor agonist. Loperamide hydrochloride is a selective and competitive Loperamide HCl
  40. BCC7003 GNTI dihydrochloride GNTI dihydrochloride
  41. BCC4612 Naloxone HCl Broad spectrum opioid antagonist,Naloxone HCl is an opioid inverse agonist drug used to counter the effects of opiate overdose. Naloxone HCl
  42. BCC1670 JDTic JDTic is a highly selective antagonist for the κ-opioid receptor; without affecting the μ- or δ-opioid receptors. JDTic
  43. BCC4615 Trimebutine Trimebutine is a drug with antimuscarinic and weak mu opioid agonist effects. Trimebutine
  44. BCC6368 Morphine hydrochloride Morphine hydrochloride
  45. BCC5215 Buprenorphine hydrochloride Buprenorphine hydrochloride
  46. BCC6093 Nalmefene - d3 Nalmefene - d3
  47. BCC5831 [Leu5]-Enkephalin [Leu5]-Enkephalin is a pentapeptides with morphine like properties. [Leu5]-Enkephalin is a five amino acid endogenous peptide that acts as an agonist at opioid receptors. [Leu5]-Enkephalin
  48. BCC7857 Nalmefene hydrochloride Nalmefene hydrochloride
  49. BCC4920 Meptazinol HCl Meptazinol is a unique centrally active opioid analgesic, which inhibits [3H]dihydromorphine binding with IC50 of 58 nM. Meptazinol HCl
  50. BCC6064 DADLE DADLE
  51. BCC6665 (±)-U-50488 hydrochloride (±)-U-50488 hydrochloride
  52. BCC6850 β-Funaltrexamine hydrochloride β-Funaltrexamine hydrochloride
  53. BCC1740 Methylnaltrexone Bromide Methylnaltrexone (Bromide) is a <b>peripheral-acting opioid receptor</b> antagonist that acts on the gastrointestinal tract to decrease opioid-induced constipation. Methylnaltrexone Bromide
  54. BCC5718 DSLET DSLET
  55. BCC5255 Oxymorphone Oxymorphone
  56. BCC5797 BAM 22P BAM-22P, a highly potent opioid peptide, is a potent opioid agonist. BAM 22P
  57. BCC6958 DAMGO DAMGO is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR. DAMGO
  58. BCC1671 JDTic 2HCl JDTic (dihydrochloride) is a potent antagonist of kappa-opioid receptors (KOR), blocking the κ-agonist U50, 488-induced antinociception. JDTic 2HCl
  59. BCC7596 Dynorphin A Dynorphin A
  60. BCC5987 Dynorphin B Dynorphin B (1-13) acts as an agonist on opioid κ-receptor. Dynorphin B
  61. BCC5864 PL 017 PL 017
  62. BCC5677 ICI 154,129 ICI 154,129
  63. BCC5875 Salvinorin A Salvinorin A
  64. BCC1265 ADL5859 HCl ADL5859 is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel. ADL5859 HCl
  65. BCC7082 FIT FIT
  66. BCC1467 Cebranopadol Cebranopadol is an analgesic NOP and opioid receptor agonist with Kis/EC50s of 0.9 nM/13 nM, 0.7 nM/1.2 nM, 2.6 nM/17 nM, 18 nM/110 nM for human NOP, MOP, KOP and delta-opioid peptide (DOP) receptor, respectively. Cebranopadol
  67. BCC6838 BNTX maleate BNTX maleate
  68. BCC6710 Naloxonazine dihydrochloride Naloxonazine dihydrochloride
  69. BCC5758 DPDPE DPDPE
  70. BCC5675 ICI 174,864 ICI 174,864
  71. BCC6000 Fentanyl citrate Fentanyl citrate

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