Products for NMDA Receptor

  1. Cat.No. Product Name Information
  2. BCC6561 (RS)-CPP (RS)-CPP
  3. BCC6986 CGS 19755 CGS 19755
  4. BCC6571 L-Cysteinesulfinic acid L-Cysteinesulfinic acid is a potent agonist at several rat metabotropic glutamate receptors (mGluRs) with pEC50s of 3.92±0.03, 4.6±0.2, 3.9±0.2, 2.7±0.2, 4.0±0.2, and 3.94±0.08 for mGluR1, mGluR5, mGluR2, mGluR4, mGluR6, and mGluR8, respectively. L-Cysteinesulfinic acid
  5. BCC7129 Remacemide hydrochloride Remacemide hydrochloride
  6. BCC6589 (S)-(-)-HA-966 (S)-(-)-HA-966
  7. BCC5946 HU 211 Dexanabinol (HU-211) is an artificially synthesized cannabinoid derivative and lacks cannabimimetic effects. Dexanabinol exhibits not only the antioxidant and neuroprotective activities in brain but also anti-inflammatory activity by inhibiting NF-κB and decreasing cytokines such as TNFα and interleukin-6, which could ensure the integrity of BBB and reduce cell apoptosis and death. Dexanabinol is widely used in head injury or stroke treatment and has been shown to be safe in animals and humans. HU 211
  8. BCC7309 PPPA PPPA
  9. BCC7087 CGP 78608 hydrochloride CGP 78608 hydrochloride is a highly potent and selective antagonist at the glycine-binding site of the NMDA receptor, with an IC50 of 6 nM. CGP 78608 acts as a potentiator of GluN1/GluN3A-mediated glycine currents, with an estimated EC50 in the low nM range (26.3 nM). Anticonvulsant activity. CGP 78608 hydrochloride
  10. BCC7308 PMPA (NMDA antagonist) PMPA (NMDA antagonist)
  11. BCC6999 D-CPP-ene D-CPP-ene
  12. BCC4160 Felbamate hydrate Felbamate hydrate (W-554 hydrate) is a potent nonsedative anticonvulsant whose clinical effect may be related to the inhibition of N-methyl-D-aspartate (NMDA) . Felbamate hydrate
  13. BCC7292 N20C hydrochloride N20C hydrochloride
  14. BCC6013 GLYX 13 Rapastinel (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator that has characteristics of a glycine site partial agonist. GLYX 13
  15. BCC7758 5,7-Dichlorokynurenic acid sodium salt 5,7-Dichlorokynurenic acid sodium salt
  16. BCC7280 Eliprodil Eliprodil(SL-820715) is a non-competitive NR2B-NMDA receptor antagonist(IC50=1 uM), less potent for NR2A- and NR2C-containing receptors(IC50> 100 uM). Eliprodil
  17. BCC4593 (-)-MK 801 (-)-Dizocilpine maleate ((-)-MK-801 maleate) is a less active (-)-enantiomer of Dizocilpine. (-)-Dizocilpine maleate is a selective and non-competitive N-methyl-D-aspartate (NMDA) receptor antagonist with a Ki of 211.7 nM. (-)-Dizocilpine maleate has antidepressant effects. (-)-MK 801
  18. BCC5888 MNI-caged-NMDA MNI-caged-NMDA
  19. BCC6292 QNZ 46 QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist (IC50 values are 3, 6, 229, and >300, >300 μM for NR2D, NR2C, NR2A, NR2B, and GluR1, respectively). QNZ 46
  20. BCC6588 (R)-(+)-HA-966 (R)-(+)-HA-966 ((+)-HA-966) is a partial agonist/antagonist of glycine site of the N-methyl-D-aspartate (NMDA) receptor complex. (R)-(+)-HA-966 selectively blocks the activation of the mesolimbic dopamine system by amphetamine. (R)-(+)-HA-966 can cross the blood-brain barrier and has the potential for neuropathic and acute pain. (R)-(+)-HA-966
  21. BCC5771 LY 233053 LY 233053
  22. BCC6581 (R)-CPP (R)-CPP
  23. BCC5977 Conantokin-T Conantokin-T
  24. BCC7078 CGP 37849 CGP 37849 is a potent, competitive and orally active N-methyl-D-aspartate (NMDA) receptor antagonist. CGP 37849 is an anticonvulsant in rodents and has antidepressant and anxiolytic-like effects. CGP 37849
  25. BCC7053 CGP 39551 CGP 39551
  26. BCC6594 N-(4-Hydroxyphenylacetyl)spermine N-(4-Hydroxyphenylacetyl)spermine
  27. BCC7753 DL-AP5 Sodium salt DL-AP5 Sodium salt
  28. BCC4059 MDL-29951 MDL-29951 is a novel glycine antagonist of NMDA receptor activation, with Ki of 0.14 μM for [3H]glycine binding in vitro and in vivo. MDL-29951
  29. BCC6592 5,7-Dichlorokynurenic acid 5,7-Dichlorokynurenic acid
  30. BCC4159 Ro 25-6981 Maleate Ro 25-6981 Maleate is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit. Ro 25-6981 Maleate
  31. BCC7655 Ro 8-4304 hydrochloride Ro 8-4304 hydrochloride
  32. BCC7508 threo Ifenprodil hemitartrate threo Ifenprodil hemitartrate
  33. BCC6984 CCMQ CCMQ
  34. BCC6602 (R)-4-Carboxyphenylglycine (R)-4-Carboxyphenylglycine
  35. BCC6892 LY 235959 LY 235959
  36. BCC6599 (RS)-(Tetrazol-5-yl)glycine (RS)-(Tetrazol-5-yl)glycine (D,L-(tetrazol-5-yl)glycine) is a highly potent and selective N-methyl-D-aspartate (NMDA) receptor agonist. (RS)-(Tetrazol-5-yl)glycine has EC50s of 99 nM, 1.7 μM for GluN1/GluN2D and GluN1/GluN2A, respectively. (RS)-(Tetrazol-5-yl)glycine induces seizure responses and Fos in mice. (RS)-(Tetrazol-5-yl)glycine
  37. BCC6774 L-689,560 L-689560 is a potent N-methyl-D-aspartate (NMDA) receptor antagonist at the GluN1 glycine binding site. L-689560 is widely used as a radiolabeled ligand in binding studies and used for study the roles of NMDA receptors in normal neurological processes as well as in diseases. L-689,560
  38. BCC6805 (2R,3S)-Chlorpheg (2R,3S)-Chlorpheg
  39. BCC6842 L-701,324 L-701324 is an orally active and long acting anticonvulsant with high affinity and selectivity for the glycine site on the NMDA receptor. L-701,324
  40. BCC6631 Arcaine sulfate Arcaine sulfate
  41. BCC6755 L-701,252 L-701,252
  42. BCC7340 Gavestinel Gavestinel
  43. BCC4158 Ro 25-6981 Ro 25-6981 is a potent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit. IC50 values are 0.009 and 52 μM for cloned receptor subunit combinations NR1C/NR2B and NR1C/NR2A respectively. Ro 25-6981
  44. BCC1939 SDZ 220-581 SDZ 220-581 is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. SDZ 220-581
  45. BCC6992 SDZ 220-040 SDZ 220-040
  46. BCC4157 SDZ 220-581 hydrochloride SDZ 220-581 hydrochloride is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. SDZ 220-581 hydrochloride
  47. BCC6730 Synthalin sulfate Synthalin sulfate
  48. BCC5982 Ketamine hydrochloride Ketamine hydrochloride
  49. BCC7369 Co 101244 hydrochloride Co 101244 hydrochloride
  50. BCC5980 Conantokin-R Conantokin-R
  51. BCC6619 (±)-1-(1,2-Diphenylethyl)piperidine maleate (±)-1-(1,2-Diphenylethyl)piperidine maleate
  52. BCC6584 ACBC ACBC
  53. BCC6688 Ifenprodil hemitartrate Ifenprodil hemitartrate
  54. BCC4904 Felbamate Felbamate (W-554) is a potent nonsedative anticonvulsant whose clinical effect may be related to the inhibition of N-methyl-D-aspartate (NMDA). Felbamate
  55. BCC6591 Ibotenic acid Ibotenic acid has agonist activity at both the N-methyl-D-aspartate (NMDA) and trans-ACPD or metabolotropic quisqualate (Qm) receptor sites. Ibotenic acid
  56. BCC7482 TCS 46b TCS 46b
  57. BCC6864 Spermine tetrahydrochloride Spermine tetrahydrochloride is an endogenous metabolite. Spermine tetrahydrochloride
  58. BCC6865 Spermidine trihydrochloride Spermidine trihydrochloride maintains cell membrane stability, increases antioxidant enzymes activities, improving photosystem II (PSII), and relevant gene expression. Spermidine trihydrochloride significantly decreases the H2O2 and O2.- contents. Spermidine trihydrochloride
  59. BCC7930 (S)-(+)-Ketamine hydrochloride (S)-(+)-Ketamine hydrochloride
  60. BCC6205 DQP 1105 DQP 1105
  61. BCC6566 cis-ACPD cis-ACPD
  62. BCC7862 CIQ CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. CIQ
  63. BCC6570 Homoquinolinic acid Homoquinolinic acid
  64. BCC6123 TCN 213 TCN 213
  65. BCC4282 Flupirtine Flupirtine(D 9998) is a selective neuronal potassium channel opener that also has NMDA receptor antagonist properties. Flupirtine
  66. BCC7234 Ro 04-5595 hydrochloride Ro 04-5595 hydrochloride
  67. BCC5918 PPDA PPDA
  68. BCC6111 TCN 237 dihydrochloride NMDA-IN-1 is a potent and NR2B-selective NMDA antagonist with Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM; no activities on NR2A, NR2C, NR2D, hERG-channel and α1-adrenergic receptor. TCN 237 dihydrochloride
  69. BCC1288 (+)-MK 801 (+)-MK 801
  70. BCC4456 Flupirtine maleate Flupirtine Maleate(D 9998) is a selective neuronal potassium channel opener that also has NMDA receptor antagonist properties. Flupirtine maleate
  71. BCC6552 DL-AP5 DL-AP5
  72. BCC4014 (+)-MK 801 Maleate Dizocilpine maleate (MK-801 maleate) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes. (+)-MK 801 Maleate
  73. BCC6551 DL-AP7 DL-AP7
  74. BCC6554 L-AP5 L-AP5
  75. BCC6553 D-AP5 D-AP5 is a NMDA receptor antagonist. D-AP5
  76. BCC5859 Norketamine hydrochloride Norketamine hydrochloride
  77. BCC6559 D-AP7 D-AP7
  78. BCC5896 MNI-caged-D-aspartate MNI-caged-D-aspartate
  79. BCC6122 TCN 201 TCN 201
  80. BCC6573 Quinolinic acid Quinolinic acid is an endogenous N-methyl-D-aspartate (NMDA) receptor agonist synthesized from L-tryptophan via the kynurenine pathway and thereby has the potential of mediating N-methyl-D-aspartate neuronal damage and dysfunction. Quinolinic acid
  81. BCC6120 Conantokin G Conantokin G

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