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Products for 5-HT Receptor

  1. Cat.No. Product Name Information
  2. BCC7218 AS 19 AS19 is a potent, selective 5-HT7 receptor agonist with an IC50 value of 0.83 nM and a Ki of 0.6 nM. AS19 is selective for 5-HT7 over 5-HT1A, 5-HT1B, 5-HT1D, and 5-HT5A receptors (Kis = 89.7 nM, 490 nM, 6.6 nM and 98.5 nM, respectively). AS19 enhances memory consolidation and reverses Scopolamine- or Dizocilpine-induced amnesia. AS 19
  3. BCC7178 Zacopride hydrochloride Zacopride hydrochloride
  4. BCC6822 MDL 11,939 MDL 11,939
  5. BCC7183 Altanserin hydrochloride Altanserin hydrochloride
  6. BCC7517 LP 12 hydrochloride LP 12 hydrochloride
  7. BCC7246 SDZ 205-557 hydrochloride SDZ 205-557 hydrochloride
  8. BCC7143 SB 206553 hydrochloride SB 206553 hydrochloride
  9. BCC7807 WAY 208466 dihydrochloride WAY 208466 dihydrochloride
  10. BCC7919 ST 1936 oxalate ST 1936 oxalate
  11. BCC5949 SB 242084 SB 242084
  12. BCC7216 SB 258585 hydrochloride SB 258585 hydrochloride
  13. BCC7056 NAS-181 NAS-181
  14. BCC5937 SB 258719 hydrochloride SB 258719 hydrochloride
  15. BCC6890 RS 16566 dihydrochloride RS 16566 dihydrochloride
  16. BCC7836 NPEC-caged-serotonin NPEC-caged-serotonin
  17. BCC7440 Fananserin Fananserin (RP 62203) is an orally bioavailable, potent and selective 5-hydroxytryptamine2 (5-HT2) receptor antagonist, with a Ki of 0.37 nM for the rat 5-HT2A receptor. Fananserin also is a selective dopamine D4 receptor antagonist, with a Ki of 2.93 nM for the human dopamine D4 receptor. Fananserin
  18. BCC5698 Methysergide maleate Methysergide maleate
  19. BCC5680 m-CPP hydrochloride m-CPP hydrochloride
  20. BCC5272 Ramosetron Hydrochloride Ramosetron Hydrochloride(YM060 Hydrochloride) is a serotonin 5-HT3 receptor antagonist for the treatment of nausea and vomiting. Ramosetron Hydrochloride
  21. BCC6202 DV 7028 hydrochloride DV 7028 hydrochloride
  22. BCC7928 BIMU 8 Potent 5-HT<sub>4</sub> receptor full agonist BIMU 8
  23. BCC5247 Sarpogrelate hydrochloride Sarpogrelate hydrochloride (MCI-9042), a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD. Sarpogrelate hydrochloride
  24. BCC7101 LY 215840 LY 215840
  25. BCC6266 LP 20 hydrochloride LP 20 hydrochloride
  26. BCC7877 MDL 100907 Volinanserin is a potent and selective antagonist of 5-HT2 receptor, with a Ki of 0.36 nM, and shows 300-fold selectivity for 5-HT2 receptor over 5-HT1c, alpha-1 and DA D2 receptors. Volinanserin has antipsychotic activity. MDL 100907
  27. BCC6994 SDZ SER 082 fumarate SDZ SER 082 fumarate
  28. BCC6877 RS 56812 hydrochloride RS 56812 hydrochloride
  29. BCC5751 SB 200646 hydrochloride SB 200646 hydrochloride
  30. BCC7019 GR 113808 GR 113808 is a potent and highly selective 5-HT4 receptor antagonist (pKb= 8.8). GR 113808 shows 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors. GR 113808
  31. BCC6678 4F 4PP oxalate 4F 4PP oxalate
  32. BCC7437 L-703,664 succinate L-703,664 succinate
  33. BCC7536 1-Methylpsilocin 1-Methylpsilocin
  34. BCC7081 GR 127935 hydrochloride GR 127935 hydrochloride
  35. BCC5752 SB 204070 SB 204070
  36. BCC6767 RS 23597-190 hydrochloride RS 23597-190 hydrochloride
  37. BCC6727 Quipazine dimaleate Quipazine dimaleate
  38. BCC7774 CP 135807 CP 135807
  39. BCC7035 SB 204741 SB 204741
  40. BCC8025 NBOH-2C-CN hydrochloride NBOH-2C-CN hydrochloride
  41. BCC6771 2-[1-(4-Piperonyl)piperazinyl]benzothiazole 2-[1-(4-Piperonyl)piperazinyl]benzothiazole
  42. BCC7285 PNU 22394 hydrochloride PNU 22394 hydrochloride
  43. BCC6913 GR 55562 dihydrochloride GR 55562 dihydrochloride
  44. BCC6915 BW 723C86 hydrochloride 5-HT<sub>2B</sub> agonist BW 723C86 hydrochloride
  45. BCC7385 Melperone hydrochloride Melperone hydrochloride
  46. BCC7164 R-96544 hydrochloride R-96544 hydrochloride
  47. BCC5694 RS 39604 hydrochloride RS 39604 hydrochloride
  48. BCC5693 RS 67333 hydrochloride RS 67333 hydrochloride
  49. BCC6878 RS 67506 hydrochloride 5-HT<sub>4</sub> partial agonist RS 67506 hydrochloride
  50. BCC7196 Ro 60-0175 fumarate Ro 60-0175 fumarate
  51. BCC7742 Donitriptan hydrochloride 5-HT<sub>1B/1D</sub> agonist Donitriptan hydrochloride
  52. BCC6697 N-Methylquipazine dimaleate N-Methylquipazine dimaleate
  53. BCC7558 LY 272015 hydrochloride LY 272015 hydrochloride
  54. BCC7856 LY 266097 hydrochloride LY 266097 hydrochloride
  55. BCC7650 BGC 20-761 High affinity 5-HT<sub>6</sub> antagonist BGC 20-761
  56. BCC6709 Metergoline Metergoline is a psychoactive drug of the ergoline chemical class which acts as a ligand for various serotonin and dopamine receptors. Metergoline
  57. BCC6976 SB 224289 hydrochloride SB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect. SB 224289 hydrochloride
  58. BCC7036 SB 228357 SB228357 is a selective, potent oral active 5-HT2C/2B receptor antagonist with pKi values of 6.9, 8.0 and 9.0 for 5-HT2A, 5-HT2B and 5-HT2C, respectively. SB228357 has antidepressant/anxiolytic effects. SB 228357
  59. BCC5679 GR 46611 GR 46611
  60. BCC7695 ML 10302 hydrochloride ML 10302 hydrochloride
  61. BCC7408 PNU 109291 PNU 109291
  62. BCC7222 PNU 142633 PNU-142633 is a high affinity, selective and orally active 5-HT1D receptor agonist with Kis of 6 nM and > 18 000 nM for human 5-HT1D receptor and human 5-HT1B receptor, respectively. PNU-142633 has anti-migraine efficacy. PNU 142633
  63. BCC7955 Tegaserod maleate Tegaserod maleate is a partial agonist of the 5-HT4 receptor; stimulates the peristaltic reflex and accelerates gastrointestinal transit. Tegaserod maleate
  64. BCC6194 AT 1015 Long-acting 5-HT<sub>2A</sub> antagonist AT 1015
  65. BCC6987 SB 216641 hydrochloride SB 216641 hydrochloride
  66. BCC7040 SB 221284 SB 221284
  67. BCC6706 Methiothepin maleate Methiothepin maleate
  68. BCC7559 LY 334370 hydrochloride LY 334370 hydrochloride
  69. BCC6035 SB 243213 dihydrochloride SB 243213 hydrochloride is an orally active, selective and high-affinity 5-hydroxytryptamine (5-HT)2C receptor antagonist with a pKi of 9.37 and a pKb of 9.8 for human 5-HT2C receptor. SB 243213 hydrochloride has improved anxiolytic profile and has the potential for schizophrenia and motor disorders. SB 243213 dihydrochloride
  70. BCC6743 3-AQC 3-AQC
  71. BCC6882 Spiperone hydrochloride Spiperone hydrochloride
  72. BCC7512 Ro 04-6790 Ro 04-6790
  73. BCC5673 SB 203186 hydrochloride SB 203186 hydrochloride
  74. BCC7718 Org 12962 hydrochloride Org 12962 hydrochloride
  75. BCC6650 m-Chlorophenylbiguanide hydrochloride m-Chlorophenylbiguanide hydrochloride
  76. BCC6291 Org 37684 Org 37684
  77. BCC7888 EMDT oxalate EMDT oxalate is a selective 5-HT EMDT oxalate
  78. BCC7838 Zotepine Zotepine
  79. BCC7660 LY 393558 LY 393558
  80. BCC6127 MS 245 oxalate MS 245 oxalate
  81. BCC7179 WAY 161503 hydrochloride WAY 161503 hydrochloride
  82. BCC5947 DOB hydrochloride DOB hydrochloride
  83. BCC7629 NPS ALX Compound 4a dihydrochloride NPS ALX Compound 4a is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist with an IC50 of 7.2 nM, which also has a great binding affinity with Ki of 0.2 nM. NPS ALX Compound 4a dihydrochloride
  84. BCC6265 PU 02 PU 02
  85. BCC7595 SB 399885 hydrochloride SB-399885 hydrochloride is a 5-HT6 receptor antagonist. SB 399885 hydrochloride
  86. BCC7990 DR 4485 hydrochloride DR 4485 hydrochloride
  87. BCC6733 MDL 72222 Bemesetron (MDL 72222) is a selective 5-HT3 receptor antagonist with an IC50 of 0.33 nM. Neuroprotective effect. MDL 72222
  88. BCC5925 DOI hydrochloride DOI hydrochloride
  89. BCC7750 SGS 518 oxalate SGS 518 oxalate
  90. BCC7562 CJ 033466 CJ 033466
  91. BCC6168 Psilocin Psilocin
  92. BCC6653 Cinanserin hydrochloride Cinanserin hydrochloride (SQ 10643) is a potent, selective and highly affinity 5-HT2 receptor antagonist with a Ki of 41 nM. Cinanserin hydrochloride has a much higher binding affinity for the 5-HT2 than for the 5-HT1 receptor (Ki of 3500 nM). Cinanserin is also an inhibitor of 3C-like proteinase of severe acute respiratory syndrome coronavirus and strongly reduces virus replication in vitro. Cinanserin hydrochloride
  93. BCC6870 1-Phenylbiguanide hydrochloride 1-Phenylbiguanide hydrochloride
  94. BCC6691 Methylergometrine maleate Methylergometrine maleate (Methylergonovine maleate) is an ergot alkaloid and an active metabolite of Methysergide with vasoconstrictive and uterotonic activity. Methylergometrine maleate is a potent, selective and orally active 5-HT receptors antagonist with a pA2 value of 9.6. Methylergometrine maleate has antimigraine and dopaminergic activity. Methylergometrine maleate can used for the prevention and control of postpartum hemorrhage. Methylergometrine maleate
  95. BCC7271 WAY 629 hydrochloride WAY 629 hydrochloride
  96. BCC6887 N-Desmethylclozapine N-Desmethylclozapine is a major active metabolite of the atypical antipsychotic drug Clozapine. N-Desmethylclozapine is a potent, allosteric and partial M1 receptors agonist (EC50=115 nM) and is able to potentiate hippocampal N-methyl-d-aspartate (NMDA) receptor currents through M1 receptor activation. N-Desmethylclozapine is also a δ-opioid agonist. N-Desmethylclozapine
  97. BCC6856 MK 212 hydrochloride MK 212 hydrochloride
  98. BCC5224 Dihydroergotamine mesylate Dihydroergotamine mesylate is an ergot alkaloid used to treat migraines. Dihydroergotamine mesylate
  99. BCC6496 Cyclobenzaprine HCl Cyclobenzaprine hydrochloride (MK130 hydrochloride) is a skeletal muscle relaxant and a central nervous system (CNS) depressant. Cyclobenzaprine HCl
  100. BCC5423 RU 24969 RU 24969 is a selective agonist at the 5-HT1A and 5-HT1B receptors. RU 24969
  101. BCC8065 Pimavanserin Pimavanserin is a selective inverse agonist of the 5-HT2A receptor with pIC50 and pKd of 8.73 and 9.3, respectively. Pimavanserin

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