GABA Receptor
GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.
Products for GABA Receptor
- Cat.No. Product Name Information
- BCN3763 (-)-Bicuculline methochloride Water-soluble GABAA antagonist
- BCN6250 Hispidulin Partial positive allosteric modulator at the benzodiazepine receptor
- BCC1327 Acamprosate calciumGlutamatergic modulator and GABA agonist
- BCC1560 EtifoxineGABAA receptor potentiator
- BCC1561 Etifoxine hydrochlorideGABAA receptor potentiator and TSPO ligand; promotes axonal regeneration
- BCC1890 Retigabine dihydrochlorideAntiepileptic compound
- BCC1940 SDZ 220-581 Ammonium saltNMDA glutamate receptor antagonist
- BCC2039 VigabatrinGABA transaminase inhibitor
- BCC4045 AWD 131-138GABAA receptor agonist
- BCC4123 (R)-Baclofen hydrochlorideGABAB receptor agonist
- BCC4255 Etomidate hydrochloride
- BCC4503 (R)-baclofen
- BCC5078 RufinamideProlongs inactivation of sodium channels; anticonvulsant
- BCC5692 SCH 50911Selective, competitive, orally active GABAB antagonist
- BCC5705 PicrotoxinGABAA receptor antagonist
- BCC5737 CGP 55845 hydrochloridePotent, selective GABAB antagonist
- BCC5957 DPNI-caged-GABANitroindoline-caged GABA
- BCC5970 LorazepamActs at the benzodiazepine modulatory site
- BCC6012 RuBi-GABACaged GABA; excitable by visible wavelength
- BCC6070 MRK 016
- BCC6087 TCS 1105
- BCC6107 FlunitrazepamActs at the benzodiazepene modulatory site
- BCC6167 OcinaplonGABAA modulator; anxiolytic
- BCC6169 TP 003
- BCC6170 MK 0343Subtype-selective GABAA receptor partial agonist
- BCC6193 PHP 501 trifluoroacetatePotent GABAA antagonist
- BCC6230 Phenobarbital sodium saltEnhances GABAergic activity
- BCC6231 Pentobarbital sodium saltEnhances GABAergic activity
- BCC6555 (-)-Bicuculline methobromideWater-soluble GABAA antagonist
- BCC6562 PhaclofenWeak, selective GABAB antagonist
- BCC6563 ZAPA sulfateAgonist at 'low affinity' GABAA receptor. More potent than GABA/muscimol
- BCC6564 TACAGABA uptake inhibitor. Also GABAA agonist and substrate for GABA-T
- BCC6574 Guvacine hydrochlorideSpecific GABA uptake inhibitor
- BCC6575 Isoguvacine hydrochlorideSelective GABAA agonist
- BCC6576 (±)-Nipecotic acidGABA uptake inhibitor
- BCC6579 2-Hydroxysaclofen
- BCC6580 SaclofenSelective GABAB antagonist
- BCC6593 MuscimolPotent GABAA agonist
- BCC6626 SKF 97541Extremely potent GABAB agonist
- BCC6629 3-Methyl-GABAActivator of GABA amino-transferase
- BCC6635 β-CCBBenzodiazepine inverse agonist, putative endogenous ligand
- BCC6671 Dihydroergotoxine mesylateBinds to GABAA receptor Cl- channel; allosteric modulator of benzodiazepine site
- BCC6685 trans-4-Hydroxycrotonic acid
- BCC6694 FG 7142Benzodiazepine inverse agonist
- BCC6738 FGIN-1-27Potent, specific ligand for mitochondrial DBI receptor
- BCC6739 FGIN-1-43Potent, specific ligand for mitochondrial DBI receptor
- BCC6745 PK 11195Antagonist at peripheral benzodiazepine receptors
- BCC6787 GBLD 345benzodiazepine receptor agonist, potent
- BCC6794 NCS-382
- BCC6803 THIP hydrochlorideGABAA agonist
- BCC6830 Chlormethiazole hydrochloridePotentiates GABAA receptor function
- BCC6903 TPMPA
- BCC6930 SKF 89976A hydrochloridePotent GABA uptake inhibitor. Penetrates blood brain barrier
- BCC6934 CGP 54626 hydrochloridePotent, selective GABAB antagonist
- BCC6988 CGP 35348Brain penetrant, selective GABAB antagonist
- BCC6989 CGP 52432Potent, selective GABAB antagonist
- BCC6990 CGP 46381Brain penetrant, selective GABAB antagonist
- BCC6997 SR 95531 hydrobromideSelective, competitive GABAA receptor antagonist
- BCC7009 Loreclezole hydrochlorideSubtype-selective GABAA receptor modulator
- BCC7010 CI 966 hydrochlorideSelective inhibitor of GAT-1
- BCC7023 L-655,708
- BCC7095 SB 205384GABAA receptor modulator; slows current decay
- BCC7096 CGP 7930Positive modulator at GABAB receptors
- BCC7097 CGP 13501Positive modulator at GABAB receptors
- BCC7115 Tracazolate hydrochlorideSubtype-selective GABAA allosteric modulator
- BCC7117 (S)-SNAP 5114GABA uptake inhibitor
- BCC7162 CL 218872Benzodiazepine agonist
- BCC7176 NNC 711Selective inhibitor of GAT-1
- BCC7186 N-ArachidonylGABAInhibits pain in vivo
- BCC7227 ZK 93423 hydrochloridePotent benzodiazepine agonist
- BCC7228 Ro 19-4603Benzodiazepine inverse agonist
- BCC7229 ZK 93426 hydrochloridePotent, competitive benzodiazepine antagonist
- BCC7230 Ro 15-4513Benzodiazepine partial inverse agonist
- BCC7233 GS 39783Positive modulator at GABAB receptors
- BCC7266 SCS
- BCC7375 CGS 20625
- BCC7387 (-)-Bicuculline methiodideWater-soluble GABAA antagonist
- BCC7397 GanaxolonePotent, positive allosteric modulator of GABAA receptors
- BCC7452 17-PAAntagonist of neurosteroid potentiation and direct gating of GABAA
- BCC7453 PentylenetetrazoleCNS stimulant
- BCC7465 U 90042GABAA receptor ligand
- BCC7466 U 89843APositive allosteric modulator of GABAA receptors
- BCC7470 Org 20599Positive allosteric modulator and direct agonist of GABAA receptors
- BCC7471 U 93631GABAA receptor antagonist
- BCC7472 NNC 05-2090 hydrochlorideGABA uptake inhibitor; moderately BGT-1 selective
- BCC7510 TB 21007
- BCC7545 AlphaxaloneDirect activator and potentiator of GABAA
- BCC7546 Valerenic acid
- BCC7560 DMCM hydrochlorideBenzodiazepine inverse agonist
- BCC7605 CGP 36216 hydrochlorideGABAB antagonist; displays activity at presynaptic receptors
- BCC7617 L-838,417Subtype-selective GABAA partial agonist
- BCC7644 rac BHFFPotent, selective GABAB positive allosteric modulator
- BCC7711 BretazenilBenzodiazepine partial agonist
- BCC7720 IndiplonSubtype-selective GABAA receptor positive allosteric modulator
- BCC7736 PregnanoloneGABAA receptor positive allosteric modulator
- BCC7737 AllopregnanoloneGABAA receptor positive allosteric modulator
- BCC7748 DS2
- BCC7819 TCS 1205Subtype-selective GABAA receptor agonist
- BCC7829 AA 29504Positive allosteric modulator of GABAA receptors