GABA Receptor
GABA receptors are a class of receptors that respond to the GABA (neurotransmitter gamma-aminobutyric acid), the chief inhibitory neurotransmitter in the vertebrate central nervous system.
Products for GABA Receptor
- Cat.No. Product Name Information
-
BCN3763
(-)-Bicuculline methochloride Water-soluble GABAA antagonist
-
BCN6250
Hispidulin Partial positive allosteric modulator at the benzodiazepine receptor
-
BCC1327
Acamprosate calciumGlutamatergic modulator and GABA agonist
-
BCC1560
EtifoxineGABAA receptor potentiator
-
BCC1561
Etifoxine hydrochlorideGABAA receptor potentiator and TSPO ligand; promotes axonal regeneration
-
BCC1890
Retigabine dihydrochlorideAntiepileptic compound
-
BCC1940
SDZ 220-581 Ammonium saltNMDA glutamate receptor antagonist
-
BCC2039
VigabatrinGABA transaminase inhibitor
-
BCC4045
AWD 131-138GABAA receptor agonist
-
BCC4123
(R)-Baclofen hydrochlorideGABAB receptor agonist
-
BCC4255
Etomidate hydrochloride
-
BCC4503
(R)-baclofen
-
BCC5078
RufinamideProlongs inactivation of sodium channels; anticonvulsant
-
BCC5692
SCH 50911Selective, competitive, orally active GABAB antagonist
-
BCC5705
PicrotoxinGABAA receptor antagonist
-
BCC5737
CGP 55845 hydrochloridePotent, selective GABAB antagonist
-
BCC5957
DPNI-caged-GABANitroindoline-caged GABA
-
BCC5970
LorazepamActs at the benzodiazepine modulatory site
-
BCC6012
RuBi-GABACaged GABA; excitable by visible wavelength
-
BCC6070
MRK 016
-
BCC6087
TCS 1105
-
BCC6107
FlunitrazepamActs at the benzodiazepene modulatory site
-
BCC6167
OcinaplonGABAA modulator; anxiolytic
-
BCC6169
TP 003
-
BCC6170
MK 0343Subtype-selective GABAA receptor partial agonist
-
BCC6193
PHP 501 trifluoroacetatePotent GABAA antagonist
-
BCC6230
Phenobarbital sodium saltEnhances GABAergic activity
-
BCC6231
Pentobarbital sodium saltEnhances GABAergic activity
-
BCC6555
(-)-Bicuculline methobromideWater-soluble GABAA antagonist
-
BCC6562
PhaclofenWeak, selective GABAB antagonist
-
BCC6563
ZAPA sulfateAgonist at 'low affinity' GABAA receptor. More potent than GABA/muscimol
-
BCC6564
TACAGABA uptake inhibitor. Also GABAA agonist and substrate for GABA-T
-
BCC6574
Guvacine hydrochlorideSpecific GABA uptake inhibitor
-
BCC6575
Isoguvacine hydrochlorideSelective GABAA agonist
-
BCC6576
(±)-Nipecotic acidGABA uptake inhibitor
-
BCC6579
2-Hydroxysaclofen
-
BCC6580
SaclofenSelective GABAB antagonist
-
BCC6593
MuscimolPotent GABAA agonist
-
BCC6626
SKF 97541Extremely potent GABAB agonist
-
BCC6629
3-Methyl-GABAActivator of GABA amino-transferase
-
BCC6635
β-CCBBenzodiazepine inverse agonist, putative endogenous ligand
-
BCC6671
Dihydroergotoxine mesylateBinds to GABAA receptor Cl- channel; allosteric modulator of benzodiazepine site
-
BCC6685
trans-4-Hydroxycrotonic acid
-
BCC6694
FG 7142Benzodiazepine inverse agonist
-
BCC6738
FGIN-1-27Potent, specific ligand for mitochondrial DBI receptor
-
BCC6739
FGIN-1-43Potent, specific ligand for mitochondrial DBI receptor
-
BCC6745
PK 11195Antagonist at peripheral benzodiazepine receptors
-
BCC6787
GBLD 345benzodiazepine receptor agonist, potent
-
BCC6794
NCS-382
-
BCC6803
THIP hydrochlorideGABAA agonist
-
BCC6830
Chlormethiazole hydrochloridePotentiates GABAA receptor function
-
BCC6903
TPMPA
-
BCC6930
SKF 89976A hydrochloridePotent GABA uptake inhibitor. Penetrates blood brain barrier
-
BCC6934
CGP 54626 hydrochloridePotent, selective GABAB antagonist
-
BCC6988
CGP 35348Brain penetrant, selective GABAB antagonist
-
BCC6989
CGP 52432Potent, selective GABAB antagonist
-
BCC6990
CGP 46381Brain penetrant, selective GABAB antagonist
-
BCC6997
SR 95531 hydrobromideSelective, competitive GABAA receptor antagonist
-
BCC7009
Loreclezole hydrochlorideSubtype-selective GABAA receptor modulator
-
BCC7010
CI 966 hydrochlorideSelective inhibitor of GAT-1
-
BCC7023
L-655,708
-
BCC7095
SB 205384GABAA receptor modulator; slows current decay
-
BCC7096
CGP 7930Positive modulator at GABAB receptors
-
BCC7097
CGP 13501Positive modulator at GABAB receptors
-
BCC7115
Tracazolate hydrochlorideSubtype-selective GABAA allosteric modulator
-
BCC7117
(S)-SNAP 5114GABA uptake inhibitor
-
BCC7162
CL 218872Benzodiazepine agonist
-
BCC7176
NNC 711Selective inhibitor of GAT-1
-
BCC7186
N-ArachidonylGABAInhibits pain in vivo
-
BCC7227
ZK 93423 hydrochloridePotent benzodiazepine agonist
-
BCC7228
Ro 19-4603Benzodiazepine inverse agonist
-
BCC7229
ZK 93426 hydrochloridePotent, competitive benzodiazepine antagonist
-
BCC7230
Ro 15-4513Benzodiazepine partial inverse agonist
-
BCC7233
GS 39783Positive modulator at GABAB receptors
-
BCC7266
SCS
-
BCC7375
CGS 20625
-
BCC7387
(-)-Bicuculline methiodideWater-soluble GABAA antagonist
-
BCC7397
GanaxolonePotent, positive allosteric modulator of GABAA receptors
-
BCC7452
17-PAAntagonist of neurosteroid potentiation and direct gating of GABAA
-
BCC7453
PentylenetetrazoleCNS stimulant
-
BCC7465
U 90042GABAA receptor ligand
-
BCC7466
U 89843APositive allosteric modulator of GABAA receptors
-
BCC7470
Org 20599Positive allosteric modulator and direct agonist of GABAA receptors
-
BCC7471
U 93631GABAA receptor antagonist
-
BCC7472
NNC 05-2090 hydrochlorideGABA uptake inhibitor; moderately BGT-1 selective
-
BCC7510
TB 21007
-
BCC7545
AlphaxaloneDirect activator and potentiator of GABAA
-
BCC7546
Valerenic acid
-
BCC7560
DMCM hydrochlorideBenzodiazepine inverse agonist
-
BCC7605
CGP 36216 hydrochlorideGABAB antagonist; displays activity at presynaptic receptors
-
BCC7617
L-838,417Subtype-selective GABAA partial agonist
-
BCC7644
rac BHFFPotent, selective GABAB positive allosteric modulator
-
BCC7711
BretazenilBenzodiazepine partial agonist
-
BCC7720
IndiplonSubtype-selective GABAA receptor positive allosteric modulator
-
BCC7736
PregnanoloneGABAA receptor positive allosteric modulator
-
BCC7737
AllopregnanoloneGABAA receptor positive allosteric modulator
-
BCC7748
DS2
-
BCC7819
TCS 1205Subtype-selective GABAA receptor agonist
-
BCC7829
AA 29504Positive allosteric modulator of GABAA receptors