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Products for GABA Receptor

  1. Cat.No. Product Name Information
  2. BCC6012 RuBi-GABA RuBi-GABA
  3. BCC6997 SR 95531 hydrobromide Gabazine is a selective and competitive antagonist of GABAA receptor, with an IC50 of ~0.2 μM for GABA receptor. SR 95531 hydrobromide
  4. BCC5078 Rufinamide Rufinamide(E 2080; CGP 33101; RUF 331) is a new antiepileptic agent that differs structurally from other antiepileptic drugs and is approved as adjunctive therapy for Lennox-Gastaut syndrome (LGS). Rufinamide
  5. BCC7010 CI 966 hydrochloride CI 966 hydrochloride
  6. BCC7375 CGS 20625 CGS 20625
  7. BCC7115 Tracazolate hydrochloride Tracazolate hydrochloride
  8. BCC6562 Phaclofen Phaclofen
  9. BCC6579 2-Hydroxysaclofen 2-Hydroxysaclofen
  10. BCC7009 Loreclezole hydrochloride Loreclezole, an antiepileptic compound, is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit containing receptors. Loreclezole hydrochloride
  11. BCC7560 DMCM hydrochloride DMCM hydrochloride is a nonselective full inverse agonist of benzodiazepine. DMCM shows bnding afinity at human recombinant GABAA αxβ3γ2 receptor subtypes with Kis of 10 nM, 13 nM, 7.5 nM, 2.2 nM for α1, α2, α3, and α5 receptors, respectively. DMCM hydrochloride
  12. BCC7227 ZK 93423 hydrochloride Potent benzodiazepine agonist ZK 93423 hydrochloride
  13. BCC7229 ZK 93426 hydrochloride ZK 93426 hydrochloride
  14. BCC6787 GBLD 345 GBLD 345
  15. BCC7644 rac BHFF rac BHFF
  16. BCC6193 PHP 501 trifluoroacetate PHP 501 trifluoroacetate
  17. BCC6988 CGP 35348 Brain penetrant, selective GABA<sub>B</sub> antagonist CGP 35348
  18. BCC6990 CGP 46381 CGP 46381
  19. BCC7605 CGP 36216 hydrochloride GABA<sub>B</sub> antagonist; displays activity at presynaptic receptors CGP 36216 hydrochloride
  20. BCC5705 Picrotoxin Picrotoxin (Cocculin) is a natural noncompetitive antagonist of GABAA receptor, binds to the interface pocket on the GABAR. Picrotoxin (Cocculin) causes overstimulation and induces convulsions. Picrotoxin
  21. BCC6580 Saclofen Saclofen
  22. BCC6626 SKF 97541 SKF 97541
  23. BCC7736 Pregnanolone Pregnanolone
  24. BCC7186 N-ArachidonylGABA N-ArachidonylGABA
  25. BCC7023 L-655,708 L-655708 is a potent α5 subunit-selective GABAA receptor inverse agonist (Ki = 0.45 nM). L-655,708
  26. BCC7465 U 90042 U 90042
  27. BCC6989 CGP 52432 CGP52432 is a GABAB receptor antagonist, with an IC50 of 85 nM. CGP 52432
  28. BCC6738 FGIN-1-27 FGIN-1-27
  29. BCN6250 Hispidulin Hispidulin is a natural flavone with a broad spectrum of biological activities. Hispidulin is a Pim-1 inhibitor with an IC50 of 2.71 μM. Hispidulin
  30. BCC6739 FGIN-1-43 FGIN-1-43
  31. BCC7176 NNC 711 NNC 711
  32. BCC6934 CGP 54626 hydrochloride CGP 54626 hydrochloride
  33. BCC5737 CGP 55845 hydrochloride Potent, selective GABA<sub>B</sub> antagonist CGP 55845 hydrochloride
  34. BCC1890 Retigabine dihydrochloride Retigabine dihydrochloride
  35. BCC7471 U 93631 U93631 is a GABAA receptor ligand of novel chemical structure with IC50 of 100 nM,and has been shown to induce a rapid, time-dependent decay of GABA-induced whole-cell Cl-currents in recombinant GABAA receptors. U 93631
  36. BCC7470 Org 20599 Org 20599
  37. BCC7466 U 89843A U 89843A
  38. BCC7117 (S)-SNAP 5114 (S)-SNAP5114 is a selective GABA transport inhibitor, with IC50 values of 5 μM and 21 μM for hGAT-3 and rGAT-2, respectively. (S)-SNAP5114 is an anticonvulsant drug. (S)-SNAP 5114
  39. BCC7095 SB 205384 GABA<sub>A</sub> receptor modulator; slows current decay SB 205384
  40. BCC6107 Flunitrazepam Flunitrazepam
  41. BCC1940 SDZ 220-581 Ammonium salt SDZ 220-581 Ammonium salt is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7. SDZ 220-581 Ammonium salt
  42. BCC6903 TPMPA TPMPA
  43. BCC7472 NNC 05-2090 hydrochloride NNC 05-2090 hydrochloride
  44. BCC6087 TCS 1105 TCS 1105
  45. BCC4045 AWD 131-138 AWD 131-138
  46. BCC7510 TB 21007 TB 21007
  47. BCC1560 Etifoxine Etifoxine(HOE 36-801) is potentiator of GABAA receptor function in cultured neurons. Etifoxine preferentially acts on β2 or β3 subunit-containing GABAA receptors. Etifoxine
  48. BCC6170 MK 0343 MK0343 (MRK-409) is an orally bioavailable GABAA receptor subtype-selective partial agonist. MK0343 is a non-sedating anxiolytic. MK 0343
  49. BCC7545 Alphaxalone Alphaxalone
  50. BCC6685 trans-4-Hydroxycrotonic acid trans-4-Hydroxycrotonic acid
  51. BCC6593 Muscimol Potent GABA<sub>A</sub> agonist Muscimol
  52. BCC7617 L-838,417 L-838,417
  53. BCC7266 SCS SCS
  54. BCC7720 Indiplon Indiplon
  55. BCC7819 TCS 1205 TCS 1205
  56. BCC7546 Valerenic acid Valerenic acid
  57. BCC6563 ZAPA sulfate ZAPA sulfate
  58. BCC7748 DS2 DS2
  59. BCC6564 TACA TACA
  60. BCC7397 Ganaxolone Ganaxolone
  61. BCC7233 GS 39783 GS 39783
  62. BCC7387 (-)-Bicuculline methiodide (-)-Bicuculline methiodide
  63. BCC7737 Allopregnanolone GABA<sub>A</sub> receptor positive allosteric modulator Allopregnanolone
  64. BCC6794 NCS-382 NCS-382
  65. BCC4255 Etomidate hydrochloride Etomidate Hcl(R16659 Hcl) is a GABAA receptors agonist, which is a short acting intravenous anaesthetic agent used for the induction of general anaesthesia. Etomidate hydrochloride
  66. BCN3763 (-)-Bicuculline methochloride (-)-Bicuculline methochloride (l-Bicuculline methochloride) is a potent GABAA receptor antagonist. (-)-Bicuculline methochloride blocks afterhyperpolarizations (AHPs) mediated by Ca2+-activated K+ channels in various types of neurons. (-)-Bicuculline methochloride
  67. BCC7453 Pentylenetetrazole Pentylenetetrazole
  68. BCC7097 CGP 13501 Positive modulator at GABA<sub>B</sub> receptors CGP 13501
  69. BCC1561 Etifoxine hydrochloride Etifoxine hydrochloride (HOE 36-801 hydrochlorid) is potentiator of GABAA receptor function in cultured neurons. Etifoxine hydrochloride
  70. BCC6230 Phenobarbital sodium salt Phenobarbital sodium salt
  71. BCC6231 Pentobarbital sodium salt Pentobarbital sodium salt
  72. BCC7096 CGP 7930 CGP 7930
  73. BCC6830 Chlormethiazole hydrochloride Chlormethiazole hydrochloride
  74. BCC6576 (±)-Nipecotic acid (±)-Nipecotic acid
  75. BCC6574 Guvacine hydrochloride Guvacine hydrochloride is an alkaloid from the nut of Areca catechu, acts as an inhibitor of GABA transporter, and dispalys modest selectivity for cloned GABA transporters with IC50s of 14 μM (human GAT-1), 39 μM (rat GAT-1), 58 μM (rat GAT-2), 119 μM (human GAT-3), 378 μM (rat GAT-3), and 1870 μM (human BGT-3). Guvacine hydrochloride
  76. BCC6169 TP 003 TP 003
  77. BCC4123 (R)-Baclofen hydrochloride (R)-Baclofen hydrochloride (STX 209 hydrochloride) is a selective GABAB receptor agonist. (R)-Baclofen hydrochloride
  78. BCC7162 CL 218872 CL 218872
  79. BCC2039 Vigabatrin Vigabatrin(γ-Vinyl-GABA; Sabril) is a structural analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that irreversibly inhibits the catabolism of GABA by GABA transaminase. Vigabatrin
  80. BCC6575 Isoguvacine hydrochloride Isoguvacine hydrochloride is a GABA receptor agonist. Isoguvacine hydrochloride
  81. BCC4503 (R)-baclofen (R)-Baclofen(STX209) is a selective GABAB receptor agonist. (R)-baclofen
  82. BCC7452 17-PA 17-PA
  83. BCC6629 3-Methyl-GABA 3-Methyl-GABA
  84. BCC5692 SCH 50911 SCH 50911, (+)-(S)-5,5-dimethylmorpholinyl-2-acetic acid, a selective, orally-active and competitive γ-Aminobutyric acid B GABA(B) receptor antagonist, binds to GABA(B) receptor with IC50 of 1.1 μM. SCH 50911 antagonizes GABA(B) autoreceptors, increasing the electrically-stimulated 3H overflow with an IC50 of 3 μM. SCH 50911
  85. BCC6555 (-)-Bicuculline methobromide (-)-Bicuculline methobromide (l-Bicuculline methobromide) is a potent GABAA receptor antagonist. (-)-Bicuculline methobromide blocks afterhyperpolarizations (AHPs) mediated by Ca2+-activated K+ channels in various types of neurons. (-)-Bicuculline methobromide
  86. BCC1327 Acamprosate calcium Acamprosate calcium(Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems; reduces alcohol consumption in animal models of alcohol addiction. Acamprosate calcium
  87. BCC6070 MRK 016 MRK 016
  88. BCC6694 FG 7142 FG 7142 (ZK 39106; LSU-65), a non-selectively benzodiazepine inverse agonist, has high affinity for the α1 subunit-containing GABAA receptor (Ki=91 nM). FG 7142 (ZK 39106; LSU-65) also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit (EC50= 137 nM). FG 7142 (ZK 39106; LSU-65) can increase tyrosine hydroxylation and cause upregulation of β-adrenoceptors in mouse cerebral cortex. FG 7142
  89. BCC6671 Dihydroergotoxine mesylate Dihydroergotoxine mesylate is a complex of closely related alkaloid salts; Binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site. Dihydroergotoxine mesylate
  90. BCC7711 Bretazenil Bretazenil
  91. BCC6635 β-CCB β-CCB
  92. BCC5970 Lorazepam Lorazepam
  93. BCC6803 THIP hydrochloride Gaboxadol hydrochloride (Lu 02-030 hydrochloride; THIP hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors (IC50=25 μM). Gaboxadol hydrochloride displays a partial agonist efficacy on subunit α1β2γ2 with an ED50 value of 143 µM, a full agonist efficacy at α5 subunit (ED50=28-129 µM) and a superagonist efficacy at α4β3δ (ED50=6 µM). Gaboxadol hydrochloride is a non-opioid analgesic and has hypnotic activities. THIP hydrochloride
  94. BCC6930 SKF 89976A hydrochloride SKF89976A hydrochloride is a selective GABA transporter (GAT-1) inhibitor with IC50s of 0.28 μM, 137.34 μM and 202.8 μM for GAT-1, GAT-2 and GAT-3 in CHO cells, respectively. SKF 89976A hydrochloride
  95. BCC6745 PK 11195 PK 11195 (RP 52028) is a ligand of translocator protein (TSPO), which targets Leishmania chemotherapy, with IC50s of 14.2 μM, 8.2 μM, 3.5 μM for L. amazonensis, L. major and L. braziliensis, respectively. PK 11195
  96. BCC7230 Ro 15-4513 Ro15-4513, imidazobenzodiazepinone derivative, is a partial inverse agonist of benzodiazepine receptor (BZR). Ro15-4513 is a potent ethanol antagonist. Ro15-4513 has anti-anxiety effect. Ro 15-4513
  97. BCC5957 DPNI-caged-GABA Nitroindoline-caged GABA DPNI-caged-GABA
  98. BCC7829 AA 29504 Positive allosteric modulator of GABA<sub>A</sub> receptors AA 29504
  99. BCC6167 Ocinaplon Ocinaplon
  100. BCC7228 Ro 19-4603 Ro 19-4603

Items 1 to 99 of 99 total

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